CYCLIC, DISULFIDE-CONTAINING AND DITHIOETHER-CONTAINING OPIOID TETRAPEPTIDES - DEVELOPMENT OF A LIGAND WITH HIGH DELTA OPIOID RECEPTOR SELECTIVITY AND AFFINITY

被引：72

作者：

MOSBERG, HI

OMNAAS, JR

MEDZIHRADSKY, F

SMITH, CB

机构：

[1] UNIV MICHIGAN,DEPT BIOL CHEM,ANN ARBOR,MI 48109

[2] UNIV MICHIGAN,DEPT PHARM,ANN ARBOR,MI 48109

来源：

LIFE SCIENCES | 1988年 / 43卷 / 12期

关键词：

D O I：

10.1016/0024-3205(88)90547-4

中图分类号：

R-3 [医学研究方法]; R3 [基础医学];

学科分类号：

1001 ;

摘要：

引用

页码：1013 / 1020

页数：8

共 15 条

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[5] [D-PEN2,L-CYS5]ENKEPHALINAMIDE AND [D-PEN2,D-CYS5]ENKEPHALINAMIDE, CONFORMATIONALLY CONSTRAINED CYCLIC ENKEPHALINAMIDE ANALOGS WITH DELTA RECEPTOR SPECIFICITY [J].

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[6]

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[8]

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[9] BIS-PENICILLAMINE ENKEPHALINS POSSESS HIGHLY IMPROVED SPECIFICITY TOWARD DELTA-OPIOID RECEPTORS [J].

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HURST, R ;

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[10]

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