STRUCTURE-ACTIVITY-RELATIONSHIPS INVOLVING THE CATECHOL SUBUNIT OF ROLIPRAM

被引：19

作者：

STAFFORD, JA

FELDMAN, PL

MARRON, BE

SCHOENEN, FJ

VALVANO, NL

UNWALLA, RJ

DOMANICO, PL

BRAWLEY, ES

LEESNITZER, MA

ROSE, DA

DOUGHERTY, RW

机构：

[1] GLAXO INC,RES INST,DEPT MOLEC SCI,RES TRIANGLE PK,NC 27709

[2] GLAXO INC,RES INST,DEPT BIOCHEM,RES TRIANGLE PK,NC 27709

[3] GLAXO INC,RES INST,DEPT CELLULAR BIOCHEM,RES TRIANGLE PK,NC 27709

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1994年 / 4卷 / 15期

关键词：

D O I：

10.1016/S0960-894X(01)80384-X

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Structure-activity relationships involving the aromatic ring of the selective PDE IV inhibitor, rolipram (1), are discussed.

引用

页码：1855 / 1860

页数：6

共 12 条

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