THE KINETICS AND DISPLACEMENT OF [FLUNITRAZEPAM-C-11 IN THE BRAIN OF THE LIVING BABOON

被引:29
作者
COMAR, D
MAZIERE, M
CEPEDA, C
GODOT, JM
MENINI, C
NAQUET, R
机构
[1] CEA, DEPT BIOL, SERV HOSP F JOLIOT, F-91191 GIF SUR YVETTE, FRANCE
[2] CNRS, DEPT NEUROPHYSIOL APPL, PHYSIOL NERVEUSE LAB, F-91190 GIF SUR YVETTE, FRANCE
关键词
D O I
10.1016/0014-2999(81)90340-X
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:21 / 26
页数:6
相关论文
共 14 条
  • [1] SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION)
    BRAESTRUP, C
    SQUIRES, RF
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) : 3805 - 3809
  • [2] BENZODIAZEPINE RECEPTORS - LABELING IN INTACT ANIMALS WITH [H-3]FLUNITRAZEPAM
    CHANG, RSL
    SNYDER, SH
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (02) : 213 - 218
  • [3] VISUALIZATION OF FLUNITRAZEPAM-C-11 DISPLACEMENT IN THE BRAIN OF THE LIVE BABOON
    COMAR, D
    MAZIERE, M
    GODOT, JM
    BERGER, G
    SOUSSALINE, F
    MENINI, C
    ARFEL, G
    NAQUET, R
    [J]. NATURE, 1979, 280 (5720) : 329 - 331
  • [4] INVIVO RECEPTOR OCCUPATION BY BENZODIAZEPINES AND CORRELATION WITH THE PHARMACOLOGICAL EFFECT
    DUKA, T
    HOLLT, V
    HERZ, A
    [J]. BRAIN RESEARCH, 1979, 179 (01) : 147 - 156
  • [5] PHARMACOKINETIC PROFILES OF CLONAZEPAM IN DOG AND HUMANS AND OF FLUNITRAZEPAM IN DOG
    KAPLAN, SA
    ALEXANDER, K
    JACK, ML
    PUGLISI, CV
    DESILVA, JAF
    LEE, TL
    WEINFELD, RE
    [J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1974, 63 (04) : 527 - 532
  • [6] MAZIERE B, 1981, J LABELLED COMPD RAD, V18, P165
  • [7] HIGH SPECIFIC ACTIVITY C-11 LABELING OF BENZODIAZEPINES - DIAZEPAM AND FLUNITRAZEPAM
    MAZIERE, M
    GODOT, JM
    BERGER, G
    PRENANT, C
    COMAR, D
    [J]. JOURNAL OF RADIOANALYTICAL CHEMISTRY, 1980, 56 (1-2): : 229 - 235
  • [8] PROPERTIES OF DIAZEPAM-H-3 BINDING TO BENZODIAZEPINE RECEPTORS IN RAT CEREBRAL-CORTEX
    MOHLER, H
    OKADA, T
    [J]. LIFE SCIENCES, 1977, 20 (12) : 2101 - 2110
  • [9] DRUGS IN BRAIN - AUTORADIOGRAPHY AND RADIOASSAY TECHNIQUES PERMIT ANALYSIS OF PENETRATION BY LABELED DRUGS
    ROTH, LJ
    BARLOW, CF
    [J]. SCIENCE, 1961, 134 (347) : 22 - &
  • [10] PHYSICAL PERFORMANCES OF A SINGLE SLICE POSITRON TOMOGRAPHIC SYSTEM AND PRELIMINARY-RESULTS IN A CLINICAL ENVIRONMENT
    SOUSSALINE, F
    TODDPOKROPEK, AE
    PLUMMER, D
    COMAR, D
    LOCH, C
    HOULE, S
    KELLERSHOHN, C
    [J]. EUROPEAN JOURNAL OF NUCLEAR MEDICINE, 1979, 4 (04): : 237 - 249