CIRCUMVENTION OF THE TUMOR MEMBRANE BARRIER TO WR-2721 ABSORPTION BY REDUCTION OF DRUG HYDROPHILICITY

被引:34
作者
YUHAS, JM
DAVIS, ME
GLOVER, D
BROWN, DQ
RITTER, M
机构
[1] UNIV PENN,DEPT HEMATOL ONCOL,PHILADELPHIA,PA 19104
[2] CHILDRENS HOSP,CHILDRENS CANC RES CTR,PHILADELPHIA,PA 19104
来源
INTERNATIONAL JOURNAL OF RADIATION ONCOLOGY BIOLOGY PHYSICS | 1982年 / 8卷 / 3-4期
关键词
D O I
10.1016/0360-3016(82)90674-5
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:519 / 522
页数:4
相关论文
共 9 条
  • [1] PARTITION-COEFFICIENT AS A GUIDE TO THE DEVELOPMENT OF RADIOSENSITIZERS WHICH ARE LESS TOXIC THAN MISONIDAZOLE
    BROWN, JM
    WORKMAN, P
    [J]. RADIATION RESEARCH, 1980, 82 (01) : 171 - 190
  • [2] GAUGAS JM, 1981, POLYAMINES NORMAL NE, P56
  • [3] KOLLMANN G, 1973, RADIAT RES, V55, P603
  • [4] INVITRO STUDIES ON THE ABSORPTION OF WR-2721 BY TUMORS AND NORMAL-TISSUES
    RITTER, MA
    BROWN, DQ
    GLOVER, DJ
    YUHAS, JM
    [J]. INTERNATIONAL JOURNAL OF RADIATION ONCOLOGY BIOLOGY PHYSICS, 1982, 8 (3-4): : 523 - 526
  • [5] DISTRIBUTION OF S-35-LABELED WR-2721 IN NORMAL AND MALIGNANT TISSUES OF MOUSE
    UTLEY, JF
    MARLOWE, C
    WADDELL, WJ
    [J]. RADIATION RESEARCH, 1976, 68 (02) : 284 - 291
  • [6] DISTRIBUTION OF WR-2721 IN NORMAL AND MALIGNANT TISSUES OF MICE AND RATS BEARING SOLID TUMORS - DEPENDENCE ON TUMOR TYPE, DRUG DOSE AND SPECIES
    WASHBURN, LC
    CARLTON, JE
    HAYES, RL
    [J]. RADIATION RESEARCH, 1974, 59 (02) : 475 - 483
  • [7] YUHAS JM, 1980, CANCER RES, V40, P1519
  • [8] PROTECTIVE DRUGS IN CANCER-THERAPY - OPTIMAL CLINICAL-TESTING AND FUTURE-DIRECTIONS
    YUHAS, JM
    [J]. INTERNATIONAL JOURNAL OF RADIATION ONCOLOGY BIOLOGY PHYSICS, 1982, 8 (3-4): : 513 - 517
  • [9] Yuhas JMS, 1980, RAD SENSITIZERS, P303