HIGH-AFFINITY INHIBITION OF [H-3-LABELED FLUNITRAZEPAM BINDING TO BRAIN BENZODIAZEPINE RECEPTORS BY CGS 9896, A NOVEL PYRAZOLOQUINOLINE

被引：11

作者：

GEE, KW

HORST, WD

OBRIEN, R

YAMAMURA, HI

机构：

[1] HOFFMANN LA ROCHE INC,DEPT PHARMACOL,NUTLEY,NJ 07110

[2] UNIV ARIZONA,ARIZONA HLTH SCI CTR,DEPT PSYCHIAT,TUCSON,AZ 85724

[3] UNIV ARIZONA,ARIZONA HLTH SCI CTR,DEPT BIOCHEM,TUCSON,AZ 85724

[4] UNIV ARIZONA,ARIZONA HLTH SCI CTR,ARIZONA RES LABS,TUCSON,AZ 85724

来源：

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | 1982年 / 105卷 / 02期

关键词：

D O I：

10.1016/0006-291X(82)91456-5

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：457 / 461

页数：5

共 11 条

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GEE KW, 1982, UNPUB LIFE SCI

[5] RESOLUTION OF 2 BIOCHEMICALLY AND PHARMACOLOGICALLY DISTINCT BENZODIAZEPINE RECEPTORS [J].

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SANO, MC ;

BEER, B .

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[6] BENZODIAZEPINE RECEPTORS - CELLULAR AND BEHAVIORAL-CHARACTERISTICS [J].

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CRITCHETT, D ;

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BEER, B .

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[7] THE PROCONVULSANT AND DIAZEPAM-REVERSING EFFECTS OF ETHYL-BETA-CARBOLINE-3-CARBOXYLATE [J].

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JONES, BJ .

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[8]

REGAN JW, 1981, MOL PHARMACOL, V20, P477

[9] SOME PROPERTIES OF BRAIN SPECIFIC BENZODIAZEPINE RECEPTORS - NEW EVIDENCE FOR MULTIPLE RECEPTORS [J].

SQUIRES, RF ;

BENSON, DI ;

BRAESTRUP, C ;

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MYERS, V ;

BEER, B .

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[10]

YAMAMURA HI, 1982, EUR J PHARM

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