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A NEW POTENTIAL PRODRUG TO IMPROVE THE DURATION OF L-DOPA - L-3-(3-HYDROXY-4-PIVALOYLOXYPHENYL)ALANINE
被引:21
作者
:
IHARA, M
论文数:
0
引用数:
0
h-index:
0
IHARA, M
TSUCHIYA, Y
论文数:
0
引用数:
0
h-index:
0
TSUCHIYA, Y
SAWASAKI, Y
论文数:
0
引用数:
0
h-index:
0
SAWASAKI, Y
HISAKA, A
论文数:
0
引用数:
0
h-index:
0
HISAKA, A
TAKEHANA, H
论文数:
0
引用数:
0
h-index:
0
TAKEHANA, H
TOMIMOTO, K
论文数:
0
引用数:
0
h-index:
0
TOMIMOTO, K
YANO, M
论文数:
0
引用数:
0
h-index:
0
YANO, M
机构
:
来源
:
JOURNAL OF PHARMACEUTICAL SCIENCES
|
1989年
/ 78卷
/ 07期
关键词
:
D O I
:
10.1002/jps.2600780703
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:525 / 529
页数:5
相关论文
共 21 条
[1]
IMPROVED DELIVERY THROUGH BIOLOGICAL-MEMBRANES .4. PRODRUGS OF L-DOPA
[J].
BODOR, N
论文数:
0
引用数:
0
h-index:
0
机构:
INTER RES CORP,LAWRENCE,KS 66044
BODOR, N
;
SLOAN, KB
论文数:
0
引用数:
0
h-index:
0
机构:
INTER RES CORP,LAWRENCE,KS 66044
SLOAN, KB
;
HIGUCHI, T
论文数:
0
引用数:
0
h-index:
0
机构:
INTER RES CORP,LAWRENCE,KS 66044
HIGUCHI, T
;
SASAHARA, K
论文数:
0
引用数:
0
h-index:
0
机构:
INTER RES CORP,LAWRENCE,KS 66044
SASAHARA, K
.
JOURNAL OF MEDICINAL CHEMISTRY,
1977,
20
(11)
:1435
-1445
[2]
CONTROLLED-RELEASE LEVODOPA CARBIDOPA .2. SINEMET CR4 TREATMENT OF RESPONSE FLUCTUATIONS IN PARKINSONS-DISEASE
[J].
CEDARBAUM, JM
论文数:
0
引用数:
0
h-index:
0
机构:
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CEDARBAUM, JM
;
BRECK, L
论文数:
0
引用数:
0
h-index:
0
机构:
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
BRECK, L
;
KUTT, H
论文数:
0
引用数:
0
h-index:
0
机构:
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
KUTT, H
;
MCDOWELL, FH
论文数:
0
引用数:
0
h-index:
0
机构:
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
MCDOWELL, FH
.
NEUROLOGY,
1987,
37
(10)
:1607
-1612
[3]
METHYLDOPAHYDRAZINE AS AN ADJUNCT TO L-DOPA THERAPY IN PARKINSONISM
[J].
CHASE, TN
论文数:
0
引用数:
0
h-index:
0
CHASE, TN
;
WATANABE, AM
论文数:
0
引用数:
0
h-index:
0
WATANABE, AM
.
NEUROLOGY,
1972,
22
(04)
:384
-&
[4]
L-DOPA ESTERS AS POTENTIAL PRODRUGS .3. BEHAVIORAL ACTIVITY IN EXPERIMENTAL-MODELS OF PARKINSONS-DISEASE
[J].
COOPER, DR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
COOPER, DR
;
MARREL, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
MARREL, C
;
VANDEWATERBEEMD, H
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
VANDEWATERBEEMD, H
;
TESTA, B
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
TESTA, B
;
JENNER, P
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
JENNER, P
;
MARSDEN, CD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
MARSDEN, CD
.
JOURNAL OF PHARMACY AND PHARMACOLOGY,
1987,
39
(08)
:627
-635
[5]
SYNTHESIS AND ANTIRESERPINE ACTIVITY OF PEPTIDES OF L-DOPA
[J].
FELIX, AM
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
FELIX, AM
;
WINTER, DP
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
WINTER, DP
;
WANG, SS
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
WANG, SS
;
KULESHA, ID
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
KULESHA, ID
;
POOL, WR
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
POOL, WR
;
HANE, DL
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
HANE, DL
;
SHEPPARD, H
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
SHEPPARD, H
.
JOURNAL OF MEDICINAL CHEMISTRY,
1974,
17
(04)
:422
-426
[6]
A LYMPHOTROPIC PRODRUG OF L-DOPA - SYNTHESIS, PHARMACOLOGICAL PROPERTIES, AND PHARMACOKINETIC BEHAVIOR OF 1,3-DIHEXADECANOYL-2-[(S)-2-AMINO-3-(3,4-DIHYDROXYPHENYL)PROPANOYL]PROPANE-1,2,3-TRIOL
[J].
GARZONABURBEH, A
论文数:
0
引用数:
0
h-index:
0
机构:
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
GARZONABURBEH, A
;
POUPAERT, JH
论文数:
0
引用数:
0
h-index:
0
机构:
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
POUPAERT, JH
;
CLAESEN, M
论文数:
0
引用数:
0
h-index:
0
机构:
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CLAESEN, M
;
DUMONT, P
论文数:
0
引用数:
0
h-index:
0
机构:
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
DUMONT, P
.
JOURNAL OF MEDICINAL CHEMISTRY,
1986,
29
(05)
:687
-691
[7]
PARKINSONS-DISEASE AND MOTOR FLUCTUATIONS - LONG-ACTING CARBIDOPA LEVODOPA (CR-4-SINEMET)
[J].
GOETZ, CG
论文数:
0
引用数:
0
h-index:
0
GOETZ, CG
;
TANNER, CM
论文数:
0
引用数:
0
h-index:
0
TANNER, CM
;
KLAWANS, HL
论文数:
0
引用数:
0
h-index:
0
KLAWANS, HL
;
SHANNON, KM
论文数:
0
引用数:
0
h-index:
0
SHANNON, KM
;
CARROLL, VS
论文数:
0
引用数:
0
h-index:
0
CARROLL, VS
.
NEUROLOGY,
1987,
37
(05)
:875
-878
[8]
GRANERUS AK, 1978, ACTA MED SCAND, V203, P75
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ON-OFF FLUCTUATIONS IN PARKINSONS-DISEASE - A CLINICAL AND NEURO-PHARMACOLOGICAL STUDY
[J].
HARDIE, RJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV COLL HOSP LONDON,DEPT NEUROL,LONDON WC1,ENGLAND
UNIV COLL HOSP LONDON,DEPT NEUROL,LONDON WC1,ENGLAND
HARDIE, RJ
;
LEES, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV COLL HOSP LONDON,DEPT NEUROL,LONDON WC1,ENGLAND
UNIV COLL HOSP LONDON,DEPT NEUROL,LONDON WC1,ENGLAND
LEES, AJ
;
STERN, GM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV COLL HOSP LONDON,DEPT NEUROL,LONDON WC1,ENGLAND
UNIV COLL HOSP LONDON,DEPT NEUROL,LONDON WC1,ENGLAND
STERN, GM
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BRAIN,
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[10]
LEVODOPA METHYL-ESTER TREATMENT OF PARKINSONS-DISEASE
[J].
JUNCOS, JL
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
JUNCOS, JL
;
MOURADIAN, MM
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
MOURADIAN, MM
;
FABBRINI, G
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
FABBRINI, G
;
SERRATI, C
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
SERRATI, C
;
CHASE, TN
论文数:
0
引用数:
0
h-index:
0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
CHASE, TN
.
NEUROLOGY,
1987,
37
(07)
:1242
-1245
←
1
2
3
→
共 21 条
[1]
IMPROVED DELIVERY THROUGH BIOLOGICAL-MEMBRANES .4. PRODRUGS OF L-DOPA
[J].
BODOR, N
论文数:
0
引用数:
0
h-index:
0
机构:
INTER RES CORP,LAWRENCE,KS 66044
BODOR, N
;
SLOAN, KB
论文数:
0
引用数:
0
h-index:
0
机构:
INTER RES CORP,LAWRENCE,KS 66044
SLOAN, KB
;
HIGUCHI, T
论文数:
0
引用数:
0
h-index:
0
机构:
INTER RES CORP,LAWRENCE,KS 66044
HIGUCHI, T
;
SASAHARA, K
论文数:
0
引用数:
0
h-index:
0
机构:
INTER RES CORP,LAWRENCE,KS 66044
SASAHARA, K
.
JOURNAL OF MEDICINAL CHEMISTRY,
1977,
20
(11)
:1435
-1445
[2]
CONTROLLED-RELEASE LEVODOPA CARBIDOPA .2. SINEMET CR4 TREATMENT OF RESPONSE FLUCTUATIONS IN PARKINSONS-DISEASE
[J].
CEDARBAUM, JM
论文数:
0
引用数:
0
h-index:
0
机构:
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CEDARBAUM, JM
;
BRECK, L
论文数:
0
引用数:
0
h-index:
0
机构:
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
BRECK, L
;
KUTT, H
论文数:
0
引用数:
0
h-index:
0
机构:
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
KUTT, H
;
MCDOWELL, FH
论文数:
0
引用数:
0
h-index:
0
机构:
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
CORNELL UNIV,MED CTR,NEW YORK HOSP,NEW YORK,NY 10021
MCDOWELL, FH
.
NEUROLOGY,
1987,
37
(10)
:1607
-1612
[3]
METHYLDOPAHYDRAZINE AS AN ADJUNCT TO L-DOPA THERAPY IN PARKINSONISM
[J].
CHASE, TN
论文数:
0
引用数:
0
h-index:
0
CHASE, TN
;
WATANABE, AM
论文数:
0
引用数:
0
h-index:
0
WATANABE, AM
.
NEUROLOGY,
1972,
22
(04)
:384
-&
[4]
L-DOPA ESTERS AS POTENTIAL PRODRUGS .3. BEHAVIORAL ACTIVITY IN EXPERIMENTAL-MODELS OF PARKINSONS-DISEASE
[J].
COOPER, DR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
COOPER, DR
;
MARREL, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
MARREL, C
;
VANDEWATERBEEMD, H
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
VANDEWATERBEEMD, H
;
TESTA, B
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
TESTA, B
;
JENNER, P
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
JENNER, P
;
MARSDEN, CD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LONDON, DEPT NEUROL, MRC, MOVEMENT DISORDERS RES GRP, LONDON SE5 8AF, ENGLAND
MARSDEN, CD
.
JOURNAL OF PHARMACY AND PHARMACOLOGY,
1987,
39
(08)
:627
-635
[5]
SYNTHESIS AND ANTIRESERPINE ACTIVITY OF PEPTIDES OF L-DOPA
[J].
FELIX, AM
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
FELIX, AM
;
WINTER, DP
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
WINTER, DP
;
WANG, SS
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
WANG, SS
;
KULESHA, ID
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
KULESHA, ID
;
POOL, WR
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
POOL, WR
;
HANE, DL
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
HANE, DL
;
SHEPPARD, H
论文数:
0
引用数:
0
h-index:
0
机构:
HOFFMAN LA ROCHE INC,DEPT CHEM RES,NUTLEY,NJ 07110
SHEPPARD, H
.
JOURNAL OF MEDICINAL CHEMISTRY,
1974,
17
(04)
:422
-426
[6]
A LYMPHOTROPIC PRODRUG OF L-DOPA - SYNTHESIS, PHARMACOLOGICAL PROPERTIES, AND PHARMACOKINETIC BEHAVIOR OF 1,3-DIHEXADECANOYL-2-[(S)-2-AMINO-3-(3,4-DIHYDROXYPHENYL)PROPANOYL]PROPANE-1,2,3-TRIOL
[J].
GARZONABURBEH, A
论文数:
0
引用数:
0
h-index:
0
机构:
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
GARZONABURBEH, A
;
POUPAERT, JH
论文数:
0
引用数:
0
h-index:
0
机构:
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
POUPAERT, JH
;
CLAESEN, M
论文数:
0
引用数:
0
h-index:
0
机构:
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CLAESEN, M
;
DUMONT, P
论文数:
0
引用数:
0
h-index:
0
机构:
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
CATHOLIC UNIV LOUVAIN,SCH PHARM,MED CHEM LAB,B-1200 BRUSSELS,BELGIUM
DUMONT, P
.
JOURNAL OF MEDICINAL CHEMISTRY,
1986,
29
(05)
:687
-691
[7]
PARKINSONS-DISEASE AND MOTOR FLUCTUATIONS - LONG-ACTING CARBIDOPA LEVODOPA (CR-4-SINEMET)
[J].
GOETZ, CG
论文数:
0
引用数:
0
h-index:
0
GOETZ, CG
;
TANNER, CM
论文数:
0
引用数:
0
h-index:
0
TANNER, CM
;
KLAWANS, HL
论文数:
0
引用数:
0
h-index:
0
KLAWANS, HL
;
SHANNON, KM
论文数:
0
引用数:
0
h-index:
0
SHANNON, KM
;
CARROLL, VS
论文数:
0
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0
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0
机构:
NINCDS,EXPTL THERAPEUT BRANCH,BLDG 10,ROOM 5C103,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
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