A NOVEL, GENERAL, TOTALLY STEREOSELECTIVE ONE-POT SYNTHESIS OF CIS-3-SUBSTITUTED 4-FORMYLAZETIDIN-2-ONES

被引：43

作者：

ALCAIDE, B

MARTINCANTALEJO, Y

PLUMET, J

RODRIGUEZLOPEZ, J

SIERRA, MA

机构：

[1] Departamento de Química Orgánica I, Facultad de Química, Universidad Complutense

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 06期

关键词：

D O I：

10.1016/S0040-4039(00)74892-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 [有机化学]; 081704 [应用化学];

摘要：

A general, totally stereoselective one-pot synthesis of cis-3-substituted-4-formylazetidin-2-ones based upon the reaction of acid chlorides and 1,4-bis-(4-methoxyphenyl)-1,4-diazabuta-1,3-diene, as synthetic equivalent of the corresponding unknown alpha-formylimine, has been developed.

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页码：803 / 806

页数：4

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