BINDING AND METABOLISM STUDIES WITH [H-3](D-ALA2,LEU5)ENKEPHALINAMIDE AND [H-3](D-ALA2,PRO5)ENKEPHALINAMIDE - EVIDENCE FOR A SELECTIVE INTERACTION OF (D-ALA2,PRO5)ENKEPHALINAMIDE WITH MU-RECEPTORS

被引：9

作者：

AUDIGIER, Y ^{[1
]}

MAZARGUIL, H ^{[1
]}

ROY, J ^{[1
]}

MORGAT, JL ^{[1
]}

CROS, J ^{[1
]}

机构：

[1] CENS, DEPT BIOL, SERV BIOCHIM, F-91191 GIF SUR YVETTE, FRANCE

来源：

EUROPEAN JOURNAL OF PHARMACOLOGY | 1981年 / 74卷 / 04期

关键词：

D O I：

10.1016/0014-2999(81)90045-5

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：273 / 278

页数：6

共 19 条

[1]

AUDIGIER Y, 1980, EUR J MED CHEM, V15, P173

[2] STRUCTURE-ACTIVITY-RELATIONSHIPS OF ENKEPHALIN ANALOGS AT OPIATE AND ENKEPHALIN RECEPTORS - CORRELATION WITH ANALGESIA [J].

AUDIGIER, Y ;

MAZARGUIL, H ;

GOUT, R ;

CROS, J .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 63 (01) :35-46

[3] OPIATE RECEPTORS IN MICE - GENETIC DIFFERENCES [J].

BARAN, A ;

SHUSTER, L ;

ELEFTHERIOU, BE ;

BAILEY, DW .

LIFE SCIENCES, 1975, 17 (04) :633-640

[4]

CRAVES FB, 1978, J PHARMACOL EXP THER, V206, P492

[5] INHIBITORY POTENCY OF VARIOUS PEPTIDES ON ENKEPHALINASE ACTIVITY FROM MOUSE STRIATUM [J].

FOURNIEZALUSKI, MC ;

PERDRISOT, R ;

GACEL, G ;

SWERTS, JP ;

ROQUES, BP ;

SCHWARTZ, JC .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 91 (01) :130-135

[6] COMPARISON OF THE BINDING CHARACTERISTICS OF TRITIATED OPIATES AND OPIOID-PEPTIDES [J].

GILLAN, MGC ;

KOSTERLITZ, HW ;

PATERSON, SJ .

BRITISH JOURNAL OF PHARMACOLOGY, 1980, 70 (03) :481-490

[7]

GILLAN MGC, 1978, CHARACTERISTICS FUNC, P475

[8] MODE OF DEACTIVATION OF ENKEPHALINS BY RAT AND HUMAN-PLASMA AND RAT-BRAIN HOMOGENATES [J].

HAMBROOK, JM ;

MORGAN, BA ;

RANCE, MJ ;

SMITH, CFC .

NATURE, 1976, 262 (5571) :782-783

[9] CHARACTERIZATION OF OPIOID RECEPTORS IN NERVOUS-TISSUE [J].

KOSTERLITZ, HW ;

PATERSON, SJ ;

MORLEY, JS .

PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1980, 210 (1178) :113-122

[10]

KOSTERLITZ HW, 1979, BRAIN PEPTIDES NEW E, P373

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