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SELECTIVITY FOR OMEGA-RECEPTOR SUBTYPES AS A STRATEGY FOR THE DEVELOPMENT OF ANXIOLYTIC DRUGS
被引:65
作者
:
LANGER, SZ
论文数:
0
引用数:
0
h-index:
0
机构:
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
LANGER, SZ
[
1
]
ARBILLA, S
论文数:
0
引用数:
0
h-index:
0
机构:
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
ARBILLA, S
[
1
]
TAN, S
论文数:
0
引用数:
0
h-index:
0
机构:
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
TAN, S
[
1
]
LLOYD, KG
论文数:
0
引用数:
0
h-index:
0
机构:
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
LLOYD, KG
[
1
]
GEORGE, P
论文数:
0
引用数:
0
h-index:
0
机构:
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
GEORGE, P
[
1
]
ALLEN, J
论文数:
0
引用数:
0
h-index:
0
机构:
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
ALLEN, J
[
1
]
WICK, AE
论文数:
0
引用数:
0
h-index:
0
机构:
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
WICK, AE
[
1
]
机构
:
[1]
SYNTHELABO LERS, DEPT CHEM, F-75621 PARIS 13, FRANCE
来源
:
PHARMACOPSYCHIATRY
|
1990年
/ 23卷
关键词
:
D O I
:
10.1055/s-2007-1014544
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
引用
收藏
页码:103 / 107
页数:5
相关论文
共 28 条
[1]
PHARMACOLOGICAL PROFILE OF THE IMIDAZOPYRIDINE ZOLPIDEM AT BENZODIAZEPINE RECEPTORS AND ELECTROCORTICOGRAM IN RATS
[J].
ARBILLA, S
论文数:
0
引用数:
0
h-index:
0
机构:
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
ARBILLA, S
;
DEPOORTERE, H
论文数:
0
引用数:
0
h-index:
0
机构:
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
DEPOORTERE, H
;
GEORGE, P
论文数:
0
引用数:
0
h-index:
0
机构:
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
GEORGE, P
;
LANGER, SZ
论文数:
0
引用数:
0
h-index:
0
机构:
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LANGER, SZ
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NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY,
1985,
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HIGH-AFFINITY [H-3] ZOLPIDEM BINDING IN THE RAT-BRAIN - AN IMIDAZOPYRIDINE WITH AGONIST PROPERTIES AT CENTRAL BENZODIAZEPINE RECEPTORS
[J].
ARBILLA, S
论文数:
0
引用数:
0
h-index:
0
机构:
LABS ETUD & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
ARBILLA, S
;
ALLEN, J
论文数:
0
引用数:
0
h-index:
0
机构:
LABS ETUD & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
ALLEN, J
;
WICK, A
论文数:
0
引用数:
0
h-index:
0
机构:
LABS ETUD & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
WICK, A
;
LANGER, SZ
论文数:
0
引用数:
0
h-index:
0
机构:
LABS ETUD & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LANGER, SZ
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1986,
130
(03)
:257
-263
[3]
BINDING OF [H-3] RO 5-4864 AND [H-3] PK 11195 TO CEREBRAL-CORTEX AND PERIPHERAL-TISSUES OF VARIOUS SPECIES - SPECIES-DIFFERENCES AND HETEROGENEITY IN PERIPHERAL BENZODIAZEPINE BINDING-SITES
[J].
AWAD, M
论文数:
0
引用数:
0
h-index:
0
机构:
TECHNION ISRAEL INST TECHNOL,FAC MED,DEPT PHARMACOL,IL-31096 HAIFA,ISRAEL
TECHNION ISRAEL INST TECHNOL,FAC MED,DEPT PHARMACOL,IL-31096 HAIFA,ISRAEL
AWAD, M
;
GAVISH, M
论文数:
0
引用数:
0
h-index:
0
机构:
TECHNION ISRAEL INST TECHNOL,FAC MED,DEPT PHARMACOL,IL-31096 HAIFA,ISRAEL
TECHNION ISRAEL INST TECHNOL,FAC MED,DEPT PHARMACOL,IL-31096 HAIFA,ISRAEL
GAVISH, M
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JOURNAL OF NEUROCHEMISTRY,
1987,
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CHARACTERIZATION OF PERIPHERAL TYPE BENZODIAZEPINE BINDING-SITES IN HUMAN AND RAT PLATELETS BY USING (H-3] PK-11195 - STUDIES IN HYPERTENSIVE PATIENTS
[J].
BENAVIDES, J
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
BENAVIDES, J
;
QUARTERONET, D
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
QUARTERONET, D
;
PLOUIN, PF
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
PLOUIN, PF
;
IMBAULT, F
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
IMBAULT, F
;
PHAN, T
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
PHAN, T
;
UZAN, A
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
UZAN, A
;
RENAULT, C
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
RENAULT, C
;
DUBROEUCQ, MC
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
DUBROEUCQ, MC
;
GUEREMY, C
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
GUEREMY, C
;
LEFUR, G
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0
引用数:
0
h-index:
0
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HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
LEFUR, G
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BIOCHEMICAL PHARMACOLOGY,
1984,
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SURICLONE - A NEW CYCLOPYRROLONE DERIVATIVE RECOGNIZING RECEPTORS LABELED BY BENZODIAZEPINES IN RAT HIPPOCAMPUS AND CEREBELLUM
[J].
BLANCHARD, JC
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BRAESTRUP, C
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AS FERROSAN,DK-2860 SOEBORG,DENMARK
BRAESTRUP, C
;
NIELSEN, M
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NIMH,BIOL PSYCHIAT BRANCH,BIOCHEM & PHARMACOL SECT,BETHESDA,MD 20014
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←
1
2
3
→
共 28 条
[1]
PHARMACOLOGICAL PROFILE OF THE IMIDAZOPYRIDINE ZOLPIDEM AT BENZODIAZEPINE RECEPTORS AND ELECTROCORTICOGRAM IN RATS
[J].
ARBILLA, S
论文数:
0
引用数:
0
h-index:
0
机构:
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
ARBILLA, S
;
DEPOORTERE, H
论文数:
0
引用数:
0
h-index:
0
机构:
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
DEPOORTERE, H
;
GEORGE, P
论文数:
0
引用数:
0
h-index:
0
机构:
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
GEORGE, P
;
LANGER, SZ
论文数:
0
引用数:
0
h-index:
0
机构:
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LAB ETUD & RECH SYNTHELABO,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LANGER, SZ
.
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY,
1985,
330
(03)
:248
-251
[2]
HIGH-AFFINITY [H-3] ZOLPIDEM BINDING IN THE RAT-BRAIN - AN IMIDAZOPYRIDINE WITH AGONIST PROPERTIES AT CENTRAL BENZODIAZEPINE RECEPTORS
[J].
ARBILLA, S
论文数:
0
引用数:
0
h-index:
0
机构:
LABS ETUD & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
ARBILLA, S
;
ALLEN, J
论文数:
0
引用数:
0
h-index:
0
机构:
LABS ETUD & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
ALLEN, J
;
WICK, A
论文数:
0
引用数:
0
h-index:
0
机构:
LABS ETUD & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
WICK, A
;
LANGER, SZ
论文数:
0
引用数:
0
h-index:
0
机构:
LABS ETUD & RECH SYNTHELABO,DEPT BIOL,58 RUE GLACIERE,F-75013 PARIS,FRANCE
LANGER, SZ
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1986,
130
(03)
:257
-263
[3]
BINDING OF [H-3] RO 5-4864 AND [H-3] PK 11195 TO CEREBRAL-CORTEX AND PERIPHERAL-TISSUES OF VARIOUS SPECIES - SPECIES-DIFFERENCES AND HETEROGENEITY IN PERIPHERAL BENZODIAZEPINE BINDING-SITES
[J].
AWAD, M
论文数:
0
引用数:
0
h-index:
0
机构:
TECHNION ISRAEL INST TECHNOL,FAC MED,DEPT PHARMACOL,IL-31096 HAIFA,ISRAEL
TECHNION ISRAEL INST TECHNOL,FAC MED,DEPT PHARMACOL,IL-31096 HAIFA,ISRAEL
AWAD, M
;
GAVISH, M
论文数:
0
引用数:
0
h-index:
0
机构:
TECHNION ISRAEL INST TECHNOL,FAC MED,DEPT PHARMACOL,IL-31096 HAIFA,ISRAEL
TECHNION ISRAEL INST TECHNOL,FAC MED,DEPT PHARMACOL,IL-31096 HAIFA,ISRAEL
GAVISH, M
.
JOURNAL OF NEUROCHEMISTRY,
1987,
49
(05)
:1407
-1414
[4]
CHARACTERIZATION OF PERIPHERAL TYPE BENZODIAZEPINE BINDING-SITES IN HUMAN AND RAT PLATELETS BY USING (H-3] PK-11195 - STUDIES IN HYPERTENSIVE PATIENTS
[J].
BENAVIDES, J
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
BENAVIDES, J
;
QUARTERONET, D
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
QUARTERONET, D
;
PLOUIN, PF
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
PLOUIN, PF
;
IMBAULT, F
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
IMBAULT, F
;
PHAN, T
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
PHAN, T
;
UZAN, A
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
UZAN, A
;
RENAULT, C
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
RENAULT, C
;
DUBROEUCQ, MC
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
DUBROEUCQ, MC
;
GUEREMY, C
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
GUEREMY, C
;
LEFUR, G
论文数:
0
引用数:
0
h-index:
0
机构:
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
HOP ST JOSEPH,SERV HYPERTENS,F-75674 PARIS,FRANCE
LEFUR, G
.
BIOCHEMICAL PHARMACOLOGY,
1984,
33
(15)
:2467
-2472
[5]
SURICLONE - A NEW CYCLOPYRROLONE DERIVATIVE RECOGNIZING RECEPTORS LABELED BY BENZODIAZEPINES IN RAT HIPPOCAMPUS AND CEREBELLUM
[J].
BLANCHARD, JC
论文数:
0
引用数:
0
h-index:
0
BLANCHARD, JC
;
JULOU, L
论文数:
0
引用数:
0
h-index:
0
JULOU, L
.
JOURNAL OF NEUROCHEMISTRY,
1983,
40
(03)
:601
-607
[6]
[H-3]-LABELED PROPYL BETA-CARBOLINE-3-CARBOXYLATE AS A SELECTIVE RADIOLIGAND FOR THE BZ1 BENZODIAZEPINE RECEPTOR SUBCLASS
[J].
BRAESTRUP, C
论文数:
0
引用数:
0
h-index:
0
机构:
AS FERROSAN,DK-2860 SOEBORG,DENMARK
BRAESTRUP, C
;
NIELSEN, M
论文数:
0
引用数:
0
h-index:
0
机构:
AS FERROSAN,DK-2860 SOEBORG,DENMARK
NIELSEN, M
.
JOURNAL OF NEUROCHEMISTRY,
1981,
37
(02)
:333
-341
[7]
INFLUENCE OF GABA RECEPTOR AGONISTS AND ANTAGONISTS ON BINDING OF DIAZEPAM-H-3 TO BENZODIAZEPINE RECEPTOR
[J].
BRILEY, MS
论文数:
0
引用数:
0
h-index:
0
BRILEY, MS
;
LANGER, SZ
论文数:
0
引用数:
0
h-index:
0
LANGER, SZ
.
EUROPEAN JOURNAL OF PHARMACOLOGY,
1978,
52
(01)
:129
-132
[8]
MOLECULAR MECHANISMS MEDIATING ACTION OF DIAZEPAM ON GABA RECEPTORS
[J].
COSTA, E
论文数:
0
引用数:
0
h-index:
0
COSTA, E
;
GUIDOTTI, A
论文数:
0
引用数:
0
h-index:
0
GUIDOTTI, A
;
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机构:
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NIMH,BIOL PSYCHIAT BRANCH,BIOCHEM & PHARMACOL SECT,BETHESDA,MD 20014
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