DO ANTIESTROGENS AND ANTIPROGESTINS ACT AS HORMONE ANTAGONISTS OR RECEPTOR-TARGETED DRUGS IN BREAST-CANCER

被引:35
作者
ROCHEFORT, H [1 ]
机构
[1] INSERM, U148, F-34100 MONTPELLIER, FRANCE
关键词
D O I
10.1016/0165-6147(87)90180-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
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收藏
页码:126 / 128
页数:3
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共 29 条
[1]   SEQUENCE-SPECIFIC DNA-BINDING OF THE PROGESTERONE-RECEPTOR TO THE UTEROGLOBIN GENE - EFFECTS OF HORMONE, ANTIHORMONE AND RECEPTOR PHOSPHORYLATION [J].
BAILLY, A ;
LEPAGE, C ;
RAUCH, M ;
MILGROM, E .
EMBO JOURNAL, 1986, 5 (12) :3235-3241
[2]   RU486, A PROGESTIN AND GLUCOCORTICOID ANTAGONIST, INHIBITS THE GROWTH OF BREAST-CANCER CELLS VIA THE PROGESTERONE-RECEPTOR [J].
BARDON, S ;
VIGNON, F ;
CHALBOS, D ;
ROCHEFORT, H .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1985, 60 (04) :692-697
[3]  
BARDON S, IN PRESS CANCER RES
[4]   INVIVO PROTEIN DNA INTERACTIONS IN A GLUCOCORTICOID RESPONSE ELEMENT REQUIRE THE PRESENCE OF THE HORMONE [J].
BECKER, PB ;
GLOSS, B ;
SCHMID, W ;
STRAHLE, U ;
SCHUTZ, G .
NATURE, 1986, 324 (6098) :686-688
[5]   PHENOL RED IN TISSUE-CULTURE MEDIA IS A WEAK ESTROGEN - IMPLICATIONS CONCERNING THE STUDY OF ESTROGEN-RESPONSIVE CELLS IN CULTURE [J].
BERTHOIS, Y ;
KATZENELLENBOGEN, JA ;
KATZENELLENBOGEN, BS .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (08) :2496-2500
[6]  
BOWEN ID, 1981, CELL DEATH BIOL PATH
[7]  
BRONZERT DA, 1985, 67TH END SOC ANN M B
[8]   A 250-KILODALTON CELLULAR PROTEIN IS INDUCED BY PROGESTINS IN 2 HUMAN-BREAST CANCER CELL-LINES MCF7 AND T47D [J].
CHALBOS, D ;
ROCHEFORT, H .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 121 (02) :421-427
[9]  
CHALBOS D, 1984, J BIOL CHEM, V259, P1231
[10]  
HERRMANN W, 1982, CR ACAD SCI III-VIE, V294, P933