NO REQUIREMENT OF CYCLIC CONFORMATION OF ANTAGONISTS IN BINDING TO VASOPRESSIN RECEPTORS

被引：88

作者：

MANNING, M ^{[1
]}

PRZYBYLSKI, JP ^{[1
]}

OLMA, A ^{[1
]}

KLIS, WA ^{[1
]}

KRUSZYNSKI, M ^{[1
]}

WO, NC ^{[1
]}

PELTON, GH ^{[1
]}

SAWYER, WH ^{[1
]}

机构：

[1] COLUMBIA UNIV COLL PHYS & SURG,DEPT PHARMACOL,NEW YORK,NY 10032

来源：

NATURE | 1987年 / 329卷 / 6142期

关键词：

D O I：

10.1038/329839a0

中图分类号：

O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];

学科分类号：

07 ; 0710 ; 09 ;

摘要：

引用

页码：839 / 840

页数：2

共 17 条

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[5] [1-BETA-MERCAPTO-BETA,BETA-DIETHYLPROPIONIC ACID]-8-LYSINE-VASOPRESSIN, A POTENT INHIBITOR OF 8-LYSINE-VASOPRESSIN AND OF OXYTOCIN [J].

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[7]

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[8] DESIGN OF MORE POTENT ANTAGONISTS OF THE ANTI-DIURETIC RESPONSES TO ARGININE-VASOPRESSIN [J].

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[9]

MANNING M, 1986, J CARDIOVASC PHAR S7, V8, P529

[10]

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