CHIRAL N-ACYLIMINIUM IONS AS NEW TOOLS IN THE ASYMMETRIC-SYNTHESIS OF CNS-ACTIVE COMPOUNDS

被引：8

作者：

WANNER, KT

机构：

[1] Institut für Pharmazie, Lebensmittelchemie der Universität München, D-80333 München

来源：

EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | 1994年 / 2卷 / 1-2期

关键词：

D O I：

10.1016/0928-0987(94)90071-X

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

[No abstract available]

引用

页码：62 / 64

页数：3

共 9 条

[1]

BEUTLER J A, 1987, Drugs of the Future, V12, P957

[2] THE ADDITION OF METALLO-ENOLATES TO CHIRAL 1-ACYLPYRIDINIUM SALTS - AN ASYMMETRIC-SYNTHESIS OF (-)-SEDAMINE [J].

COMINS, DL ;

HONG, H .

JOURNAL OF ORGANIC CHEMISTRY, 1993, 58 (19) :5035-5036

[3] PHENCYCLIDINE-LIKE EFFECTS OF TETRAHYDROISOQUINOLINES AND RELATED-COMPOUNDS [J].

GRAY, NM ;

CHENG, BK ;

MICK, SJ ;

LAIR, CM ;

CONTRERAS, PC .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (06) :1242-1248

[4] NEWER METHODS OF PREPARATIVE INORGANIC CHEMISTRY II .8. AMIDOMETHYLATIONS [J].

HELLMANN, H .

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 1957, 69 (13-4) :463-471

[5] STEREOSELECTIVE NUCLEOPHILIC-SUBSTITUTION OF 6-METHOXY-1-METHOXYCARBONYLPIPECOLATE - ENANTIOSELECTIVE SYNTHESIS OF (+)-SEDAMINE FROM L-LYSINE [J].

IRIE, K ;

AOE, K ;

TANAKA, T ;

SAITO, S .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1985, (10) :633-635

[6]

KIGUCHI T, 1990, HETEROCYCLES, V31, P1525

[7] ASYMMETRIC ALPHA-AMIDOALKYLATION - SYNTHESES OF ENANTIOMERICALLY PURE ALPHA-SUBSTITUTED PIPERIDINES WITH 1-CAMPHANOYL-1,2,3,4-TETRAHYDROPY-RIDINE [J].

WANNER, KT ;

KARTNER, A .

ARCHIV DER PHARMAZIE, 1987, 320 (12) :1253-1267

[8] ASYMMETRIC ELECTROPHILIC ALPHA-AMIDOALKYLATION .10. A NEW CAMPHORIMIDE DERIVED CHIRAL AUXILIARY FOR THE ASYMMETRIC-SYNTHESIS WITH N-ACYLIMINIUM IONS - PREPARATION OF ARACEMIC 2-SUBSTITUTED PIPERIDINES [J].

WANNER, KT ;

PAINTNER, FF .

TETRAHEDRON, 1994, 50 (10) :3113-3122

[9] THE ANTICONVULSANT MK-801 IS A POTENT N-METHYL-D-ASPARTATE ANTAGONIST [J].

WONG, EHF ;

KEMP, JA ;

PRIESTLEY, T ;

KNIGHT, AR ;

WOODRUFF, GN ;

IVERSEN, LL .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (18) :7104-7108

← 1 →