ERRORS IN THE MEASUREMENT OF AGONIST POTENCY-RATIOS PRODUCED BY UPTAKE PROCESSES - A GENERAL-MODEL APPLIED TO BETA-ADRENOCEPTOR AGONISTS

被引:39
作者
KENAKIN, TP
机构
关键词
D O I
10.1111/j.1476-5381.1980.tb10953.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:407 / 417
页数:11
相关论文
共 26 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[3]   EXTRANEURONAL REMOVAL, ACCUMULATION AND O-METHYLATION OF ISOPRENALINE IN PERFUSED HEART [J].
BONISCH, H ;
TRENDELENBURG, U .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1974, 283 (02) :191-218
[4]  
BRIMIJOIN S, 1970, J PHARMACOL EXP THER, V175, P503
[5]   INHIBITION OF NORADRENALINE UPTAKE BY SYMPATHOMIMETIC AMINES IN RAT ISOLATED HEART [J].
BURGEN, ASV ;
IVERSEN, LL .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1965, 25 (01) :34-&
[6]   ROLE OF UPTAKE OF NORADRENALINE FOR ITS POSITIVE INOTROPIC EFFECT IN RELATION TO MUSCLE GEOMETRY - STATISTICAL EVALUATION [J].
EBNER, F ;
WAUD, DR .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1978, 303 (01) :1-6
[7]   POTENTIATION OF RESPENSES TO NORA-DRENALINE AND ISOPRENALINE OF GUINEA-PIG ISOLATED TRACHEAL CHAIN PREPARATION BY DESIPRAMINE COCAINE PHENTOLAMINE PHENOXYBENZAMINE GUANETHIDINE METANEPHRINE AND COOLING [J].
FOSTER, RW .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1967, 31 (03) :466-&
[9]  
FURCHGOTT RF, 1975, FED PROC, V34, P794
[10]  
FURCHGOTT RF, 1975, 6TH INT C PHARM HELS, P622