SYNTHESIS OF A NEW MOLECULAR CARRIER - N-(LEU-ENKEPHALIN)YL 6-AMIDO-6-DEOXY-CYCLOMALTOHEPTAOSE

被引：55

作者：

DJEDAINIPILARD, F

DESALOS, J

PERLY, B

机构：

[1] Service de Chimie Moléculaire. Centre d'Etudes de Saclay.

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 15期

关键词：

D O I：

10.1016/S0040-4039(00)60440-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of N-(Leu-enkephalin)yl 6-amido-6-deoxy-cyclomaltoheptaose has been performed in high yield. The final derivative has been characterized by proton NMR in terms of chemical structure and inclusion properties and represents a new class of target-directed transporters.

引用

页码：2457 / 2460

页数：4

共 14 条

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