PROTEIN CRYSTALLOGRAPHY AND COMPUTER-GRAPHICS TOWARD RATIONAL DRUG DESIGN

被引:97
作者
HOL, WGJ
机构
来源
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH | 1986年 / 25卷 / 09期
关键词
D O I
10.1002/anie.198607673
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
收藏
页码:767 / 778
页数:12
相关论文
共 140 条
[1]   PHYSIOLOGICAL AND X-RAY STUDIES OF POTENTIAL ANTISICKLING AGENTS [J].
ABRAHAM, DJ ;
PERUTZ, MF ;
PHILLIPS, SEV .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (02) :324-328
[2]  
ABRAHAM EP, SPEKTRUM WISS 1981, P46
[3]  
ABRAHAM EP, 1981, SCI AM, V244, P64
[4]   ON THE 3-DIMENSIONAL STRUCTURE AND CATALYTIC MECHANISM OF TRIOSE PHOSPHATE ISOMERASE [J].
ALBER, T ;
BANNER, DW ;
BLOOMER, AC ;
PETSKO, GA ;
PHILLIPS, D ;
RIVERS, PS ;
WILSON, IA .
PHILOSOPHICAL TRANSACTIONS OF THE ROYAL SOCIETY OF LONDON SERIES B-BIOLOGICAL SCIENCES, 1981, 293 (1063) :159-171
[5]   X-RAY-DIFFRACTION STUDY OF BINDING OF 2,3-DIPHOSPHOGLYCERATE TO HUMAN DEOXYHEMOGLOBIN [J].
ARNONE, A .
NATURE, 1972, 237 (5351) :146-&
[6]   3-DIMENSIONAL STRUCTURE OF CALMODULIN [J].
BABU, YS ;
SACK, JS ;
GREENHOUGH, TJ ;
BUGG, CE ;
MEANS, AR ;
COOK, WJ .
NATURE, 1985, 315 (6014) :37-40
[7]   SUBSTITUTED BENZALDEHYDES DESIGNED TO INCREASE THE OXYGEN-AFFINITY OF HUMAN-HEMOGLOBIN AND INHIBIT THE SICKLING OF SICKLE ERYTHROCYTES [J].
BEDDELL, CR ;
GOODFORD, PJ ;
KNEEN, G ;
WHITE, RD ;
WILKINSON, S ;
WOOTTON, R .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 82 (02) :397-407
[8]   COMPOUNDS DESIGNED TO FIT A SITE OF KNOWN STRUCTURE IN HUMAN HEMOGLOBIN [J].
BEDDELL, CR ;
GOODFORD, PJ ;
NORRINGTON, FE ;
WILKINSON, S ;
WOOTTON, R .
BRITISH JOURNAL OF PHARMACOLOGY, 1976, 57 (02) :201-209
[9]   A H-1-NMR STUDY OF THE INTERACTIONS AND CONFORMATIONS OF RATIONALLY DESIGNED BRODIMOPRIM ANALOGS IN COMPLEXES WITH LACTOBACILLUS-CASEI DIHYDROFOLATE-REDUCTASE [J].
BIRDSALL, B ;
FEENEY, J ;
PASCUAL, C ;
ROBERTS, GCK ;
KOMPIS, I ;
THEN, RL ;
MULLER, K ;
KROEHN, A .
JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (12) :1672-1676
[10]   PHOSPHOGLYCERATE KINASE [J].
BLAKE, CCF ;
RICE, DW .
PHILOSOPHICAL TRANSACTIONS OF THE ROYAL SOCIETY OF LONDON SERIES B-BIOLOGICAL SCIENCES, 1981, 293 (1063) :93-104