H-3-(-)-BUPRANOLOL, A NEW BETA-ADRENOCEPTOR RADIOLIGAND - CHARACTERIZATION OF ITS BINDING TO KITTEN HEART BETA-ADRENOCEPTORS

被引：21

作者：

MORRIS, TH

SANDROCK, K

KAUMANN, AJ

机构：

[1] UNIV DUSSELDORF,INST PHYSIOL,LEHRSTUHL KLIN PHYSIOL,D-4000 DUSSELDORF 1,FED REP GER

[2] SANOL SCHWARZ GMBH,CHEM ABT,D-4019 MONHEIM,FED REP GER

来源：

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY | 1981年 / 317卷 / 01期

关键词：

D O I：

10.1007/BF00506251

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：19 / 25

页数：7

共 34 条

[11] IN KITTEN VENTRICULAR MYOCARDIUM, THE INOTROPIC POTENCY OF AN AGONIST IS DETERMINED BY BOTH ITS INTRINSIC ACTIVITY FOR THE ADENYLYL CYCLASE AND ITS AFFINITY FOR THE BETA-ADRENOCEPTORS [J].

KAUMANN, AJ .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1981, 317 (01) :13-18

[12] COMPARISON OF THE INFLUENCE OF N-ISOPROPYL AND N-TERT BUTYL SUBSTITUENTS ON THE AFFINITY OF LIGANDS FOR SINOATRIAL BETA-ADRENOCEPTORS IN RAT ATRIA AND BETA-ADRENOCEPTORS COUPLED TO THE ADENYLYL CYCLASE IN KITTEN VENTRICLE [J].

KAUMANN, AJ ;

MORRIS, TH ;

BIRNBAUMER, L .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 307 (01) :1-8

[13]

KAUMANN AJ, 1974, J BIOL CHEM, V249, P7874

[14] BETA-ADRENOCEPTOR BLOCKING-AGENTS AS PARTIAL AGONISTS IN ISOLATED HEART-MUSCLE - DISSOCIATION OF STIMULATION AND BLOCKADE [J].

KAUMANN, AJ ;

BLINKS, JR .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 311 (03) :237-248

[15] STIMULANT AND DEPRESSANT EFFECTS OF BETA-ADRENOCEPTOR BLOCKING-AGENTS ON ISOLATED HEART-MUSCLE - A POSITIVE INOTROPIC EFFECT NOT MEDIATED THROUGH ADRENOCEPTORS [J].

KAUMANN, AJ ;

BLINKS, JR .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 311 (03) :205-218

[16] COMPARATIVE-ASSESSMENT OF BETA-ADRENOCEPTOR BLOCKING-AGENTS AS SIMPLE COMPETITIVE ANTAGONISTS IN ISOLATED HEART-MUSCLE - SIMILARITY OF INOTROPIC AND CHRONOTROPIC BLOCKING POTENCIES AGAINST ISOPROTERENOL [J].

KAUMANN, AJ ;

MCINERNY, TK ;

GILMOUR, DP ;

BLINKS, JR .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 311 (03) :219-236

[17]

KAUMANN AJ, 1975, N-S ARCH PHARMACOL, V287, P23

[18] RELAXATION OF HEART-MUSCLE BY CATECHOLAMINES AND BY DIBUTYRYL CYCLIC ADENOSINE-3',5'-MONOPHOSPHATE - SIMILARITY OF BETA-ADRENOCEPTORS MEDIATING CONTRACTILE AND RELAXANT EFFECTS OF CATECHOLAMINES IN KITTEN PAPILLARY-MUSCLE [J].

KAUMANN, AJ .

NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1977, 296 (03) :205-215

[19]

KAUMANN AJ, 1981, NAUNYNSCHMIEDEBERGS, V315, pR59

[20] STEREOSPECIFIC [H-3] (-)-ALPRENOLOL BINDING-SITES, BETA-ADRENERGIC RECEPTORS AND ADENYLATE CYCLASE [J].

LEFKOWITZ, RJ ;

MUKHERJEE, C ;

COVERSTONE, M ;

CARON, MG .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1974, 60 (02) :703-709

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