RECENT ADVANCES IN THE SYNTHESIS OF ANTIBACTERIAL QUINOLONES

被引：58

作者：

RADL, S ^{[1
]}

BOUZARD, D ^{[1
]}

机构：

[1] BRISTOL MYERS SQUIBB,F-77200 TORCY,FRANCE

来源：

HETEROCYCLES | 1992年 / 34卷 / 11期

关键词：

D O I：

10.3987/REV-92-446

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

This review surveys the main synthetic approaches used for the construction of antibacterial quinolones, including aza analogs (naphthyridones, cinnolones) and condensed polycyclic analogs, with an emphasis on the more versatile methods which are potentially useful in other fields of heterocyclic chemistry. Simpler non-condensed monocyclic analogs, i.e., pyridone and pyridazinone carboxylic acids are also briefly mentioned.

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页码：2143 / 2177

页数：35

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