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ENZYME-INHIBITION AS A SOURCE OF NEW DRUGS
被引:15
作者
:
KALMAN, TI
论文数:
0
引用数:
0
h-index:
0
机构:
SUNY BUFFALO,SCH PHARM,DEPT BIOCHEM PHARMACOL,AMHERST,NY 14260
SUNY BUFFALO,SCH PHARM,DEPT BIOCHEM PHARMACOL,AMHERST,NY 14260
KALMAN, TI
[
1
]
机构
:
[1]
SUNY BUFFALO,SCH PHARM,DEPT BIOCHEM PHARMACOL,AMHERST,NY 14260
来源
:
DRUG DEVELOPMENT RESEARCH
|
1981年
/ 1卷
/ 04期
关键词
:
D O I
:
10.1002/ddr.430010404
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:311 / 328
页数:18
相关论文
共 53 条
[1]
SUICIDE ENZYME INACTIVATORS
ABELES, RH
论文数:
0
引用数:
0
h-index:
0
机构:
BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02154
ABELES, RH
MAYCOCK, AL
论文数:
0
引用数:
0
h-index:
0
机构:
BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02154
MAYCOCK, AL
[J].
ACCOUNTS OF CHEMICAL RESEARCH,
1976,
9
(09)
: 313
-
319
[2]
ABELES RH, 1978, ENZYME ACTIVATED IRR, P1
[3]
Baker BR, 1967, DESIGN ACTIVE SITE D
[4]
AMINO-ACID SEQUENCE AT FDUMP BINDING-SITE OF THYMIDYLATE SYNTHETASE
BELLISARIO, RL
论文数:
0
引用数:
0
h-index:
0
机构:
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
BELLISARIO, RL
MALEY, GF
论文数:
0
引用数:
0
h-index:
0
机构:
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
MALEY, GF
GALIVAN, JH
论文数:
0
引用数:
0
h-index:
0
机构:
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
GALIVAN, JH
MALEY, F
论文数:
0
引用数:
0
h-index:
0
机构:
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
MALEY, F
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1976,
73
(06)
: 1848
-
1852
[5]
BENDER ML, 1971, MECHANISMS HOMOGENEO
[6]
ON THE MECHANISM OF ACTION OF FOLATE-REQUIRING AND BIOPTERIN-REQUIRING ENZYMES
BENKOVIC, SJ
论文数:
0
引用数:
0
h-index:
0
BENKOVIC, SJ
[J].
ANNUAL REVIEW OF BIOCHEMISTRY,
1980,
49
: 227
-
251
[7]
BENKOVIC SJ, 1973, PROGR BIOORG CHEM, V2, P133
[8]
CHARACTERIZATION OF A DISTINCT MEMBRANE-BOUND DIPEPTIDYL CARBOXYPEPTIDASE INACTIVATING ENKEPHALIN IN BRAIN
BENUCK, M
论文数:
0
引用数:
0
h-index:
0
BENUCK, M
MARKS, N
论文数:
0
引用数:
0
h-index:
0
MARKS, N
[J].
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1980,
95
(02)
: 822
-
828
[9]
INHIBITION OF TESTOSTERONE 5-ALPHA-REDUCTASE BY A PROPOSED ENZYME-ACTIVATED, ACTIVE SITE-DIRECTED INHIBITOR
BLOHM, TR
论文数:
0
引用数:
0
h-index:
0
BLOHM, TR
METCALF, BW
论文数:
0
引用数:
0
h-index:
0
METCALF, BW
LAUGHLIN, ME
论文数:
0
引用数:
0
h-index:
0
LAUGHLIN, ME
SJOERDSMA, A
论文数:
0
引用数:
0
h-index:
0
SJOERDSMA, A
SCHATZMAN, GL
论文数:
0
引用数:
0
h-index:
0
SCHATZMAN, GL
[J].
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1980,
95
(01)
: 273
-
280
[10]
BOBEK M, 1978, CHEM BIOL NUCLEOSIDE, P135
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1
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6
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共 53 条
[1]
SUICIDE ENZYME INACTIVATORS
ABELES, RH
论文数:
0
引用数:
0
h-index:
0
机构:
BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02154
ABELES, RH
MAYCOCK, AL
论文数:
0
引用数:
0
h-index:
0
机构:
BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02154
MAYCOCK, AL
[J].
ACCOUNTS OF CHEMICAL RESEARCH,
1976,
9
(09)
: 313
-
319
[2]
ABELES RH, 1978, ENZYME ACTIVATED IRR, P1
[3]
Baker BR, 1967, DESIGN ACTIVE SITE D
[4]
AMINO-ACID SEQUENCE AT FDUMP BINDING-SITE OF THYMIDYLATE SYNTHETASE
BELLISARIO, RL
论文数:
0
引用数:
0
h-index:
0
机构:
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
BELLISARIO, RL
MALEY, GF
论文数:
0
引用数:
0
h-index:
0
机构:
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
MALEY, GF
GALIVAN, JH
论文数:
0
引用数:
0
h-index:
0
机构:
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
GALIVAN, JH
MALEY, F
论文数:
0
引用数:
0
h-index:
0
机构:
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
NEW YORK STATE DEPT HLTH,DIV LABS & RES,ALBANY,NY 12201
MALEY, F
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1976,
73
(06)
: 1848
-
1852
[5]
BENDER ML, 1971, MECHANISMS HOMOGENEO
[6]
ON THE MECHANISM OF ACTION OF FOLATE-REQUIRING AND BIOPTERIN-REQUIRING ENZYMES
BENKOVIC, SJ
论文数:
0
引用数:
0
h-index:
0
BENKOVIC, SJ
[J].
ANNUAL REVIEW OF BIOCHEMISTRY,
1980,
49
: 227
-
251
[7]
BENKOVIC SJ, 1973, PROGR BIOORG CHEM, V2, P133
[8]
CHARACTERIZATION OF A DISTINCT MEMBRANE-BOUND DIPEPTIDYL CARBOXYPEPTIDASE INACTIVATING ENKEPHALIN IN BRAIN
BENUCK, M
论文数:
0
引用数:
0
h-index:
0
BENUCK, M
MARKS, N
论文数:
0
引用数:
0
h-index:
0
MARKS, N
[J].
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1980,
95
(02)
: 822
-
828
[9]
INHIBITION OF TESTOSTERONE 5-ALPHA-REDUCTASE BY A PROPOSED ENZYME-ACTIVATED, ACTIVE SITE-DIRECTED INHIBITOR
BLOHM, TR
论文数:
0
引用数:
0
h-index:
0
BLOHM, TR
METCALF, BW
论文数:
0
引用数:
0
h-index:
0
METCALF, BW
LAUGHLIN, ME
论文数:
0
引用数:
0
h-index:
0
LAUGHLIN, ME
SJOERDSMA, A
论文数:
0
引用数:
0
h-index:
0
SJOERDSMA, A
SCHATZMAN, GL
论文数:
0
引用数:
0
h-index:
0
SCHATZMAN, GL
[J].
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1980,
95
(01)
: 273
-
280
[10]
BOBEK M, 1978, CHEM BIOL NUCLEOSIDE, P135
←
1
2
3
4
5
6
→