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INHIBITION OF TESTOSTERONE 5-ALPHA-REDUCTASE BY A PROPOSED ENZYME-ACTIVATED, ACTIVE SITE-DIRECTED INHIBITOR
被引:52
作者
:
BLOHM, TR
论文数:
0
引用数:
0
h-index:
0
BLOHM, TR
METCALF, BW
论文数:
0
引用数:
0
h-index:
0
METCALF, BW
LAUGHLIN, ME
论文数:
0
引用数:
0
h-index:
0
LAUGHLIN, ME
SJOERDSMA, A
论文数:
0
引用数:
0
h-index:
0
SJOERDSMA, A
SCHATZMAN, GL
论文数:
0
引用数:
0
h-index:
0
SCHATZMAN, GL
机构
:
来源
:
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
|
1980年
/ 95卷
/ 01期
关键词
:
D O I
:
10.1016/0006-291X(80)90735-4
中图分类号
:
Q5 [生物化学];
Q7 [分子生物学];
学科分类号
:
071010 ;
081704 ;
摘要
:
引用
收藏
页码:273 / 280
页数:8
相关论文
共 29 条
[1]
SUICIDE ENZYME INACTIVATORS
ABELES, RH
论文数:
0
引用数:
0
h-index:
0
机构:
BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02154
ABELES, RH
MAYCOCK, AL
论文数:
0
引用数:
0
h-index:
0
机构:
BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02154
MAYCOCK, AL
[J].
ACCOUNTS OF CHEMICAL RESEARCH,
1976,
9
(09)
: 313
-
319
[2]
ROLE OF RECEPTOR PROTEINS IN CONTROLLING ANDROGEN ACTION IN SEBACEOUS GLANDS OF HAMSTERS
ADACHI, K
论文数:
0
引用数:
0
h-index:
0
ADACHI, K
KANO, M
论文数:
0
引用数:
0
h-index:
0
KANO, M
[J].
STEROIDS,
1972,
19
(04)
: 567
-
&
[3]
[Anonymous], 1870, COMMUNICATION
[4]
BENSON HD, 1978, Patent No. 4088760
[5]
ANDROGEN METABOLISM IN ADIPOSE-TISSUE - CONVERSION OF 5ALPHA-DIHYDROTESTOSTERONE TO 3-ALPHA-ANDROSTANEDIOL BY HAMSTER TISSUE
BLOHM, TR
论文数:
0
引用数:
0
h-index:
0
BLOHM, TR
LAUGHLIN, ME
论文数:
0
引用数:
0
h-index:
0
LAUGHLIN, ME
[J].
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY,
1978,
9
(07)
: 603
-
608
[6]
BRUCHOVSKY N, 1968, J BIOL CHEM, V243, P2012
[7]
TESTOSTERONE 5ALPHA-REDUCTASE AND THE ACCUMULATION OF DIHYDROTESTOSTERONE IN BENIGN PROSTATIC HYPERPLASIA
COWAN, RA
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
COWAN, RA
COOK, B
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
COOK, B
COWAN, SK
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
COWAN, SK
GRANT, JK
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
GRANT, JK
SIRETT, DAN
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
SIRETT, DAN
WALLACE, AM
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
WALLACE, AM
[J].
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY,
1979,
11
(01)
: 609
-
613
[8]
STEROIDAL INHIBITORS OF PROSTATIC 5-ALPHA-REDUCTASE - STRUCTURE-ACTIVITY-RELATIONSHIPS
DUPUY, GM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,DEPT OBSTET & GYNECOL,MONTREAL 101,QUEBEC,CANADA
DUPUY, GM
ROBERTS, KD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,DEPT OBSTET & GYNECOL,MONTREAL 101,QUEBEC,CANADA
ROBERTS, KD
BLEAU, G
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,DEPT OBSTET & GYNECOL,MONTREAL 101,QUEBEC,CANADA
BLEAU, G
CHAPDELAINE, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,DEPT OBSTET & GYNECOL,MONTREAL 101,QUEBEC,CANADA
CHAPDELAINE, A
[J].
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY,
1978,
9
(11)
: 1043
-
1047
[9]
FREDERIKSEN DW, 1971, J BIOL CHEM, V246, P2584
[10]
A COMPARATIVE STUDY OF CONVERSION OF TESTOSTERONE TO 17BETA-HYDROXY-5ALPHA-ANDROSTAN-3-ONE (DIHYDROTESTOSTERONE) BY PROSTATE AND EPIDIDYMIS
GLOYNA, RE
论文数:
0
引用数:
0
h-index:
0
GLOYNA, RE
WILSON, JD
论文数:
0
引用数:
0
h-index:
0
WILSON, JD
[J].
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM,
1969,
29
(07)
: 970
-
+
←
1
2
3
→
共 29 条
[1]
SUICIDE ENZYME INACTIVATORS
ABELES, RH
论文数:
0
引用数:
0
h-index:
0
机构:
BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02154
ABELES, RH
MAYCOCK, AL
论文数:
0
引用数:
0
h-index:
0
机构:
BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02154
MAYCOCK, AL
[J].
ACCOUNTS OF CHEMICAL RESEARCH,
1976,
9
(09)
: 313
-
319
[2]
ROLE OF RECEPTOR PROTEINS IN CONTROLLING ANDROGEN ACTION IN SEBACEOUS GLANDS OF HAMSTERS
ADACHI, K
论文数:
0
引用数:
0
h-index:
0
ADACHI, K
KANO, M
论文数:
0
引用数:
0
h-index:
0
KANO, M
[J].
STEROIDS,
1972,
19
(04)
: 567
-
&
[3]
[Anonymous], 1870, COMMUNICATION
[4]
BENSON HD, 1978, Patent No. 4088760
[5]
ANDROGEN METABOLISM IN ADIPOSE-TISSUE - CONVERSION OF 5ALPHA-DIHYDROTESTOSTERONE TO 3-ALPHA-ANDROSTANEDIOL BY HAMSTER TISSUE
BLOHM, TR
论文数:
0
引用数:
0
h-index:
0
BLOHM, TR
LAUGHLIN, ME
论文数:
0
引用数:
0
h-index:
0
LAUGHLIN, ME
[J].
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY,
1978,
9
(07)
: 603
-
608
[6]
BRUCHOVSKY N, 1968, J BIOL CHEM, V243, P2012
[7]
TESTOSTERONE 5ALPHA-REDUCTASE AND THE ACCUMULATION OF DIHYDROTESTOSTERONE IN BENIGN PROSTATIC HYPERPLASIA
COWAN, RA
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
COWAN, RA
COOK, B
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
COOK, B
COWAN, SK
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
COWAN, SK
GRANT, JK
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
GRANT, JK
SIRETT, DAN
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
SIRETT, DAN
WALLACE, AM
论文数:
0
引用数:
0
h-index:
0
机构:
University Department of Pathological Biochemistry, Royal Infirmary, Glasgow
WALLACE, AM
[J].
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY,
1979,
11
(01)
: 609
-
613
[8]
STEROIDAL INHIBITORS OF PROSTATIC 5-ALPHA-REDUCTASE - STRUCTURE-ACTIVITY-RELATIONSHIPS
DUPUY, GM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,DEPT OBSTET & GYNECOL,MONTREAL 101,QUEBEC,CANADA
DUPUY, GM
ROBERTS, KD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,DEPT OBSTET & GYNECOL,MONTREAL 101,QUEBEC,CANADA
ROBERTS, KD
BLEAU, G
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,DEPT OBSTET & GYNECOL,MONTREAL 101,QUEBEC,CANADA
BLEAU, G
CHAPDELAINE, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MONTREAL,DEPT OBSTET & GYNECOL,MONTREAL 101,QUEBEC,CANADA
CHAPDELAINE, A
[J].
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY,
1978,
9
(11)
: 1043
-
1047
[9]
FREDERIKSEN DW, 1971, J BIOL CHEM, V246, P2584
[10]
A COMPARATIVE STUDY OF CONVERSION OF TESTOSTERONE TO 17BETA-HYDROXY-5ALPHA-ANDROSTAN-3-ONE (DIHYDROTESTOSTERONE) BY PROSTATE AND EPIDIDYMIS
GLOYNA, RE
论文数:
0
引用数:
0
h-index:
0
GLOYNA, RE
WILSON, JD
论文数:
0
引用数:
0
h-index:
0
WILSON, JD
[J].
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM,
1969,
29
(07)
: 970
-
+
←
1
2
3
→