THE REACTION OF AROMATIC ALPHA-BETA-UNSATURATED KETONES WITH 4,5-DIAMINO-1,6-DIHYDROPYRIMIDIN-6-ONES

被引：28

作者：

INSUASTY, B

RAMOS, M

QUIROGA, J

SANCHEZ, A

NOGUERAS, M

HANOLD, N

MEIER, H

机构：

[1] UNIV LOS ANDES, DEPT CHEM, BOGOTA, COLOMBIA

[2] UNIV GRANADA, COLEGIO UNIV JAEN, DEPT CHEM, E-23071 JAEN, SPAIN

[3] UNIV MAINZ, INST ORGAN CHEM, D-55099 MAINZ, GERMANY

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1994年 / 31卷 / 01期

关键词：

D O I：

10.1002/jhet.5570310111

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The reaction of 4,5-diamino-1,6-dihydropyrimidin-6-ones 1 with one equivalent of the chalcones 2 leads in an acidic medium to the formation of the 2,4-diaryl-2,3,6,7-tetrahydro-1H-pyrimido[4,5-b][l,4]diazepin-ones 3a-m. The structure elucidation of the products is based on detailed nmr investigations including selective C-13{H-1} decoupling experiments.

引用

页码：61 / 64

页数：4

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