BIARYL SYNTHESIS VIA SUZUKI COUPLING ON A SOLID SUPPORT

被引：160

作者：

FRENETTE, R ^{[1
]}

FRIESEN, RW ^{[1
]}

机构：

[1] MERCK FROSST CTR THERAPEUT RES,DEPT MED CHEM,POINTE CLAIRE H9R 4P8,PQ,CANADA

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 49期

关键词：

D O I：

10.1016/0040-4039(94)88458-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Aryl boronic acids undergo a facile and efficient palladium catalyzed cross-coupling reaction with aryl bromides and iodides that are bound to a Merrifield resin. Simple transesterification releases the biaryl products from the solid support in excellent purity and yield.

引用

页码：9177 / 9180

页数：4

共 21 条

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