A GENERAL AND EXPEDIENT METHOD FOR THE SOLID-PHASE SYNTHESIS OF 1,4-BENZODIAZEPINE DERIVATIVES

被引：426

作者：

BUNIN, BA ^{[1
]}

ELLMAN, JA ^{[1
]}

机构：

[1] UNIV CALIF BERKELEY,DEPT CHEM,BERKELEY,CA 94720

来源：

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY | 1992年 / 114卷 / 27期

关键词：

D O I：

10.1021/ja00053a067

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：10997 / 10998

页数：2

共 17 条

[1]

BORANY G, 1980, PEPTIDES, V2, P1

[2]

CAMPS F, 1974, AN QUIM, V70, P848

[3] ((9-FLUORENYLMETHYL)OXY)CARBONYL (FMOC) AMINO-ACID FLUORIDES - CONVENIENT NEW PEPTIDE COUPLING REAGENTS APPLICABLE TO THE FMOC/TERT-BUTYL STRATEGY FOR SOLUTION AND SOLID-PHASE SYNTHESES [J].

CARPINO, LA ;

SADATAALAEE, D ;

CHAO, HG ;

DESELMS, RH .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1990, 112 (26) :9651-9652

[4] NUCLEOTIDE CHEMISTRY .8. SYNTHESIS OF OLIGODEOXYNUCLEOTIDES AND OLIGODEOXYNUCLEOTIDE ANALOGS USING PHOSPHORAMIDITE INTERMEDIATES [J].

DORMAN, MA ;

NOBLE, SA ;

MCBRIDE, LJ ;

CARUTHERS, MH .

TETRAHEDRON, 1984, 40 (01) :95-102

[5] METHODS FOR DRUG DISCOVERY - DEVELOPMENT OF POTENT, SELECTIVE, ORALLY EFFECTIVE CHOLECYSTOKININ ANTAGONISTS [J].

EVANS, BE ;

RITTLE, KE ;

BOCK, MG ;

DIPARDO, RM ;

FREIDINGER, RM ;

WHITTER, WL ;

LUNDELL, GF ;

VEBER, DF ;

ANDERSON, PS ;

CHANG, RSL ;

LOTTI, VJ ;

CERINO, DJ ;

CHEN, TB ;

KLING, PJ ;

KUNKEL, KA ;

SPRINGER, JP ;

HIRSHFIELD, J .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (12) :2235-2246

[6] THE ASYMMETRIC-SYNTHESIS OF ALPHA-AMINO-ACIDS - ELECTROPHILIC AZIDATION OF CHIRAL IMIDE ENOLATES, A PRACTICAL APPROACH TO THE SYNTHESIS OF (R)-ALPHA-AZIDO AND (S)-ALPHA-AZIDO CARBOXYLIC-ACIDS [J].

EVANS, DA ;

BRITTON, TC ;

ELLMAN, JA ;

DOROW, RL .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1990, 112 (10) :4011-4030

[7] LIGHT-DIRECTED, SPATIALLY ADDRESSABLE PARALLEL CHEMICAL SYNTHESIS [J].

FODOR, SPA ;

READ, JL ;

PIRRUNG, MC ;

STRYER, L ;

LU, AT ;

SOLAS, D .

SCIENCE, 1991, 251 (4995) :767-773

[8] GENERATION AND USE OF SYNTHETIC PEPTIDE COMBINATORIAL LIBRARIES FOR BASIC RESEARCH AND DRUG DISCOVERY [J].

HOUGHTEN, RA ;

PINILLA, C ;

BLONDELLE, SE ;

APPEL, JR ;

DOOLEY, CT ;

CUERVO, JH .

NATURE, 1991, 354 (6348) :84-86

[9] INHIBITION OF HIV REPLICATION IN ACUTE AND CHRONIC INFECTIONS INVITRO BY A TAT ANTAGONIST [J].

HSU, MC ;

SCHUTT, AD ;

HOLLY, M ;

SLICE, LW ;

SHERMAN, MI ;

RICHMAN, DD ;

POTASH, MJ ;

VOLSKY, DJ .

SCIENCE, 1991, 254 (5039) :1799-1802

[10] MULTIPLE PEPTIDE-SYNTHESIS METHODS AND THEIR APPLICATIONS [J].

JUNG, G ;

BECKSICKINGER, AG .

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 1992, 31 (04) :367-383

← 1 2 →