TRICYCLIC BETA-LACTAMS - TOTAL SYNTHESIS AND ANTIBACTERIAL ACTIVITY OF 5-ALPHA-METHOXY-TRIBACTAMS AND 5-BETA-METHOXY-TRIBACTAMS

被引：18

作者：

HANESSIAN, S

ROZEMA, MJ

REDDY, GB

BRAGANZA, JF

机构：

[1] Department of Chemistry, Montréal, Que. H3C 3J7, Universite Montreal P.O. Box 6128, Succ. Centre-ville

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1995年 / 5卷 / 21期

基金：

加拿大自然科学与工程研究理事会;

关键词：

D O I：

10.1016/0960-894X(95)00445-Y

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The total synthesis of the tricyclic beta-lactams, ''5 alpha- and 5 beta-methoxy tribactams'', positional isomers of the Glare 4a-methoxy-tribactam is described and preliminary biological evaluation is reported.

引用

页码：2535 / 2540

页数：6

共 41 条

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