MOLECULAR-STRUCTURES OF 8-CHLORO-6-PHENYL-4H-S-TRIAZOLO[4,3-A][1,4]BENZODIAZEPINE, 2-ACETOXYAMINO-4-ACETYL-8-CHLORO-3,4-DIHYDRO-6-PHENYL-1,4,5-BENZOTRIAZOCINE AND 8-CHLORO-4,11-DIACETYL-4,11-DIHYDRO-2-METHYL-6-PHENYLOXAZOLO[4,5-B]-[1,4,5]BENZOTRIAZOCINE - FORMATION OF AN 8-MEMBERED RING FROM A QUINAZOLINE DERIVATIVE ON TREATMENT WITH HYDRAZINE EVIDENCED BY X-RAY ANALYSISE

被引：25

作者：

KAMIYA, K ^{[1
]}

WADA, Y ^{[1
]}

NISHIKAWA, M ^{[1
]}

机构：

[1] TAKEDA CHEM IND LTD, CENT RES DIV, HIGASHIYODOGAWA, TOKYO, JAPAN

来源：

CHEMICAL & PHARMACEUTICAL BULLETIN | 1973年 / 21卷 / 07期

关键词：

D O I：

10.1248/cpb.21.1520

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1520 / 1529

页数：10

共 12 条

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[2] DIPHENYLHYDANTOIN AND DIAZEPAM - MOLECULAR STRUCTURE SIMILARITIES AND STERIC BASIS OF ANTICONVULSANT ACTIVITY
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[3] QUINAZOLINES AND 1,4-BENZODIAZEPINES .38. REACTION OF HYDRAZINES WITH 6-CHLORO-2-CHLOROMETHYL-4-PHENYLQUINAZOLINE 3-OXIDE
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[4] CRYSTAL AND MOLECULAR STRUCTURE OF 7-CHLORO-5-(2,4-DICHLOROPHENYL)-4,5-DIHYDRO-1,4-DIMETHYL-3H-1,4-BENZODIAZEPIN-2-ONE, C17H15CL3N2O
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[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1967, 89 (04) : 804 - &
[5] MEGURO K, 1970, TETRAHEDRON LETT, P4039
[6] MEGURO K, TO BE PUBLISHED
[7] STRUCTURE-ACTIVITY RELATIONSHIP OF S-TRIAZOLO-1,4-BENZODIAZEPINES IN CENTRAL NERVOUS DEPRESSANT ACTION
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[J]. JAPANESE JOURNAL OF PHARMACOLOGY, 1971, 21 (04) : 489 - &
[8] PHARMACOLOGICAL STUDIES ON NEW POTENT CENTRAL DEPRESSANTS, 8-CHLORO-6-PHENYL-4H-S-TRIAZOLO [4,3A] [1,4] BENZODIAZEPINE (D-40TA) AND ITS 1-METHYL ANALOGUE (D-65MT)
NAKAJIMA, R
TAKE, Y
MORIYA, R
SAJI, Y
YUI, T
NAGAWA, Y
[J]. JAPANESE JOURNAL OF PHARMACOLOGY, 1971, 21 (04) : 497 - &
[9] X-RAY ANALYSES OF ACUTUMINE AND ITS ACETATE - A TRIAL OF A SHORT CUT IN STRUCTURE ELUCIDATION
NISHIKAWA, M
KAMIYA, K
TOMITA, M
OKAMOTO, Y
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OSAKI, K
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