A NEW CLASS OF NONPEPTIDIC CHOLECYSTOKININ-B GASTRIN RECEPTOR ANTAGONISTS BASED ON DIBENZOBICYCLO[2.2.2]OCTANE

被引：19

作者：

KALINDJIAN, SB

BODKIN, MJ

BUCK, IM

DUNSTONE, DJ

LOW, CMR

MCDONALD, IM

PETHER, MJ

STEEL, KIM

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1994年 / 37卷 / 22期

关键词：

D O I：

10.1021/jm00048a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：3671 / 3673

页数：3

共 18 条

[11] 2-NAPHTHALENESULPHONYL L-ASPARTYL-(2-PHENETHYL)AMIDE (2-NAP) - A SELECTIVE CHOLECYSTOKININ CCK(A)-RECEPTOR ANTAGONIST [J].

HULL, RAD ;

SHANKLEY, NP ;

HARPER, EA ;

GERSKOWITCH, VP ;

BLACK, JW .

BRITISH JOURNAL OF PHARMACOLOGY, 1993, 108 (03) :734-740

[12]

MARTINEZ J, 1986, INT J PEPT PROT RES, V28, P529

[13] STRUCTURE - FUNCTION RELATIONSHIPS IN GASTRIN-LIKE PEPTIDES [J].

MORLEY, JS .

PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1968, 170 (1018) :97-+

[14] FUNCTIONAL COMPARISONS OF GASTRIN CHOLECYSTOKININ RECEPTORS IN ISOLATED PREPARATIONS OF GASTRIC-MUCOSA AND ILEUM [J].

PATEL, M ;

SPRAGGS, CF .

BRITISH JOURNAL OF PHARMACOLOGY, 1992, 106 (02) :275-282

[15] CHOLECYSTOKININ TYPE-B RECEPTOR ANTAGONIST PD-136,450 IS A PARTIAL SECRETORY AGONIST IN THE STOMACH AND A FULL AGONIST IN THE PANCREAS OF THE RAT [J].

SCHMASSMANN, A ;

GARNER, A ;

FLOGERZI, B ;

HASAN, MY ;

SANNER, M ;

VARGA, L ;

HALTER, F .

GUT, 1994, 35 (02) :270-274

[16]

SHANKLEY NP, COMMUNICATION

[17] COMPARATIVE-ANALYSIS OF THE VAGAL-STIMULATION OF GASTRIC-ACID SECRETION IN RODENT ISOLATED STOMACH PREPARATIONS [J].

WELSH, NJ ;

SHANKLEY, NP ;

BLACK, JW .

BRITISH JOURNAL OF PHARMACOLOGY, 1994, 112 (01) :93-96

[18]

YU MJ, 1991, J MED CHEM, V34, P1508

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