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ATOMIC-STRUCTURE OF THE RAPAMYCIN HUMAN IMMUNOPHILIN FKBP-12 COMPLEX
被引:180
作者
:
VANDUYNE, GD
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
VANDUYNE, GD
STANDAERT, RF
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
STANDAERT, RF
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SCHREIBER, SL
CLARDY, J
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
CLARDY, J
机构
:
[1]
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
[2]
CORNELL UNIV,DEPT CHEM,ITHACA,NY 14853
来源
:
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
|
1991年
/ 113卷
/ 19期
关键词
:
D O I
:
10.1021/ja00019a057
中图分类号
:
O6 [化学];
学科分类号
:
0703 ;
摘要
:
[No abstract available]
引用
收藏
页码:7433 / 7434
页数:2
相关论文
共 14 条
[1]
SUBSTRATE-SPECIFICITY FOR THE HUMAN ROTAMASE FKBP - A VIEW OF FK506 AND RAPAMYCIN AS LEUCINE (TWISTED AMIDE) PROLINE MIMICS
ALBERS, MW
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
ALBERS, MW
WALSH, CT
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
WALSH, CT
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SCHREIBER, SL
[J].
JOURNAL OF ORGANIC CHEMISTRY,
1990,
55
(17)
: 4984
-
4986
[2]
PROBING IMMUNOSUPPRESSANT ACTION WITH A NONNATURAL IMMUNOPHILIN LIGAND
BIERER, BE
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
BIERER, BE
SOMERS, PK
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SOMERS, PK
WANDLESS, TJ
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
WANDLESS, TJ
BURAKOFF, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
BURAKOFF, SJ
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SCHREIBER, SL
[J].
SCIENCE,
1990,
250
(4980)
: 556
-
559
[3]
2 DISTINCT SIGNAL TRANSMISSION PATHWAYS IN LYMPHOCYTES-T ARE INHIBITED BY COMPLEXES FORMED BETWEEN AN IMMUNOPHILIN AND EITHER FK506 OR RAPAMYCIN
BIERER, BE
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
BIERER, BE
MATTILA, PS
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
MATTILA, PS
STANDAERT, RF
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
STANDAERT, RF
HERZENBERG, LA
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
HERZENBERG, LA
BURAKOFF, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
BURAKOFF, SJ
CRABTREE, G
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
CRABTREE, G
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
SCHREIBER, SL
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1990,
87
(23)
: 9231
-
9235
[4]
BRUNGER AT, 1990, XPLOR MANUAL VERSION
[5]
ON THE CHEMISTRY AND HIGH-FIELD NUCLEAR MAGNETIC-RESONANCE SPECTROSCOPY OF RAPAMYCIN
FINDLAY, JA
论文数:
0
引用数:
0
h-index:
0
机构:
CENT RES INST CHEM,NMR LAB,H-1525 BUDAPEST,HUNGARY
CENT RES INST CHEM,NMR LAB,H-1525 BUDAPEST,HUNGARY
FINDLAY, JA
RADICS, L
论文数:
0
引用数:
0
h-index:
0
机构:
CENT RES INST CHEM,NMR LAB,H-1525 BUDAPEST,HUNGARY
CENT RES INST CHEM,NMR LAB,H-1525 BUDAPEST,HUNGARY
RADICS, L
[J].
CANADIAN JOURNAL OF CHEMISTRY-REVUE CANADIENNE DE CHIMIE,
1980,
58
(06):
: 579
-
590
[6]
MERLOT, AN INTEGRATED PACKAGE OF COMPUTER-PROGRAMS FOR THE DETERMINATION OF CRYSTAL-STRUCTURES BY MOLECULAR REPLACEMENT
FITZGERALD, PMD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT BIOCHEM,EDMONTON T6G 2H7,ALBERTA,CANADA
UNIV ALBERTA,DEPT BIOCHEM,EDMONTON T6G 2H7,ALBERTA,CANADA
FITZGERALD, PMD
[J].
JOURNAL OF APPLIED CRYSTALLOGRAPHY,
1988,
21
(03)
: 273
-
278
[7]
A RECEPTOR FOR THE IMMUNOSUPPRESSANT FK506 IS A CIS-TRANS PEPTIDYL-PROLYL ISOMERASE
HARDING, MW
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARDING, MW
GALAT, A
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
GALAT, A
UEHLING, DE
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
UEHLING, DE
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SCHREIBER, SL
[J].
NATURE,
1989,
341
(6244)
: 758
-
760
[8]
RAPAMYCIN SENSITIVITY IN SACCHAROMYCES-CEREVISIAE IS MEDIATED BY A PEPTIDYL-PROLYL CIS-TRANS ISOMERASE RELATED TO HUMAN FK506-BINDING PROTEIN
KOLTIN, Y
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
KOLTIN, Y
FAUCETTE, L
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
FAUCETTE, L
BERGSMA, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
BERGSMA, DJ
LEVY, MA
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
LEVY, MA
CAFFERKEY, R
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
CAFFERKEY, R
KOSER, PL
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
KOSER, PL
JOHNSON, RK
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
JOHNSON, RK
LIVI, GP
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
LIVI, GP
[J].
MOLECULAR AND CELLULAR BIOLOGY,
1991,
11
(03)
: 1718
-
1723
[9]
SOLUTION STRUCTURE OF FKBP, A ROTAMASE ENZYME AND RECEPTOR FOR FK506 AND RAPAMYCIN
MICHNICK, SW
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
MICHNICK, SW
ROSEN, MK
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
ROSEN, MK
WANDLESS, TJ
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
WANDLESS, TJ
KARPLUS, M
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
KARPLUS, M
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SCHREIBER, SL
[J].
SCIENCE,
1991,
252
(5007)
: 836
-
839
[10]
SOLUTION STRUCTURE OF THE MAJOR BINDING-PROTEIN FOR THE IMMUNOSUPPRESSANT FK506
MOORE, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Vertex Pharmaceuticals Incorporated, Cambridge, MA 02139-4211
MOORE, JM
PEATTIE, DA
论文数:
0
引用数:
0
h-index:
0
机构:
Vertex Pharmaceuticals Incorporated, Cambridge, MA 02139-4211
PEATTIE, DA
FITZGIBBON, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
Vertex Pharmaceuticals Incorporated, Cambridge, MA 02139-4211
FITZGIBBON, MJ
THOMSON, JA
论文数:
0
引用数:
0
h-index:
0
机构:
Vertex Pharmaceuticals Incorporated, Cambridge, MA 02139-4211
THOMSON, JA
[J].
NATURE,
1991,
351
(6323)
: 248
-
250
←
1
2
→
共 14 条
[1]
SUBSTRATE-SPECIFICITY FOR THE HUMAN ROTAMASE FKBP - A VIEW OF FK506 AND RAPAMYCIN AS LEUCINE (TWISTED AMIDE) PROLINE MIMICS
ALBERS, MW
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
ALBERS, MW
WALSH, CT
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
WALSH, CT
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SCHREIBER, SL
[J].
JOURNAL OF ORGANIC CHEMISTRY,
1990,
55
(17)
: 4984
-
4986
[2]
PROBING IMMUNOSUPPRESSANT ACTION WITH A NONNATURAL IMMUNOPHILIN LIGAND
BIERER, BE
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
BIERER, BE
SOMERS, PK
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SOMERS, PK
WANDLESS, TJ
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
WANDLESS, TJ
BURAKOFF, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
BURAKOFF, SJ
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SCHREIBER, SL
[J].
SCIENCE,
1990,
250
(4980)
: 556
-
559
[3]
2 DISTINCT SIGNAL TRANSMISSION PATHWAYS IN LYMPHOCYTES-T ARE INHIBITED BY COMPLEXES FORMED BETWEEN AN IMMUNOPHILIN AND EITHER FK506 OR RAPAMYCIN
BIERER, BE
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
BIERER, BE
MATTILA, PS
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
MATTILA, PS
STANDAERT, RF
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
STANDAERT, RF
HERZENBERG, LA
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
HERZENBERG, LA
BURAKOFF, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
BURAKOFF, SJ
CRABTREE, G
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
CRABTREE, G
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
BRIGHAM & WOMENS HOSP,DEPT MED,DIV HEMATOL,BOSTON,MA 02115
SCHREIBER, SL
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1990,
87
(23)
: 9231
-
9235
[4]
BRUNGER AT, 1990, XPLOR MANUAL VERSION
[5]
ON THE CHEMISTRY AND HIGH-FIELD NUCLEAR MAGNETIC-RESONANCE SPECTROSCOPY OF RAPAMYCIN
FINDLAY, JA
论文数:
0
引用数:
0
h-index:
0
机构:
CENT RES INST CHEM,NMR LAB,H-1525 BUDAPEST,HUNGARY
CENT RES INST CHEM,NMR LAB,H-1525 BUDAPEST,HUNGARY
FINDLAY, JA
RADICS, L
论文数:
0
引用数:
0
h-index:
0
机构:
CENT RES INST CHEM,NMR LAB,H-1525 BUDAPEST,HUNGARY
CENT RES INST CHEM,NMR LAB,H-1525 BUDAPEST,HUNGARY
RADICS, L
[J].
CANADIAN JOURNAL OF CHEMISTRY-REVUE CANADIENNE DE CHIMIE,
1980,
58
(06):
: 579
-
590
[6]
MERLOT, AN INTEGRATED PACKAGE OF COMPUTER-PROGRAMS FOR THE DETERMINATION OF CRYSTAL-STRUCTURES BY MOLECULAR REPLACEMENT
FITZGERALD, PMD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ALBERTA,DEPT BIOCHEM,EDMONTON T6G 2H7,ALBERTA,CANADA
UNIV ALBERTA,DEPT BIOCHEM,EDMONTON T6G 2H7,ALBERTA,CANADA
FITZGERALD, PMD
[J].
JOURNAL OF APPLIED CRYSTALLOGRAPHY,
1988,
21
(03)
: 273
-
278
[7]
A RECEPTOR FOR THE IMMUNOSUPPRESSANT FK506 IS A CIS-TRANS PEPTIDYL-PROLYL ISOMERASE
HARDING, MW
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARDING, MW
GALAT, A
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
GALAT, A
UEHLING, DE
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
UEHLING, DE
SCHREIBER, SL
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
SCHREIBER, SL
[J].
NATURE,
1989,
341
(6244)
: 758
-
760
[8]
RAPAMYCIN SENSITIVITY IN SACCHAROMYCES-CEREVISIAE IS MEDIATED BY A PEPTIDYL-PROLYL CIS-TRANS ISOMERASE RELATED TO HUMAN FK506-BINDING PROTEIN
KOLTIN, Y
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
KOLTIN, Y
FAUCETTE, L
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
FAUCETTE, L
BERGSMA, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
BERGSMA, DJ
LEVY, MA
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
LEVY, MA
CAFFERKEY, R
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
CAFFERKEY, R
KOSER, PL
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
KOSER, PL
JOHNSON, RK
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
JOHNSON, RK
LIVI, GP
论文数:
0
引用数:
0
h-index:
0
机构:
SMITHKLINE BEECHAM PHARMACEUT,DEPT BIOMOLEC DISCOVERY,KING OF PRUSSIA,PA 19406
LIVI, GP
[J].
MOLECULAR AND CELLULAR BIOLOGY,
1991,
11
(03)
: 1718
-
1723
[9]
SOLUTION STRUCTURE OF FKBP, A ROTAMASE ENZYME AND RECEPTOR FOR FK506 AND RAPAMYCIN
MICHNICK, SW
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
MICHNICK, SW
ROSEN, MK
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
ROSEN, MK
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HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
WANDLESS, TJ
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HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
KARPLUS, M
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HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
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Vertex Pharmaceuticals Incorporated, Cambridge, MA 02139-4211
FITZGIBBON, MJ
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