EFFECTS OF THE PUTATIVE ANTAGONISTS PHACLOFEN AND DELTA-AMINOVALERIC ACID ON GABAB RECEPTOR BIOCHEMISTRY

被引：30

作者：

ROBINSON, TN ^{[1
]}

CROSS, AJ ^{[1
]}

GREEN, AR ^{[1
]}

TOCZEK, JM ^{[1
]}

BOAR, BR ^{[1
]}

机构：

[1] ASTRA NEUROSCI RES UNIT,1 WAKEFIELD ST,LONDON WC1N 1PJ,ENGLAND

来源：

BRITISH JOURNAL OF PHARMACOLOGY | 1989年 / 98卷 / 03期

关键词：

D O I：

10.1111/j.1476-5381.1989.tb14612.x

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：833 / 840

页数：8

共 31 条

[1] EVIDENCE THAT ANTAGONISM BY DELTA-AMINOVALERIC ACID OF GABA-B RECEPTORS IN THE GUINEA-PIG ILEUM MAY BE DUE TO AN INTERACTION BETWEEN GABA-A AND GABA-B RECEPTORS [J].

ALLAN, RD ;

DICKENSON, HW .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 120 (01) :119-122

[2] CHARACTERISTICS OF GABAB RECEPTOR-BINDING SITES ON RAT WHOLE BRAIN SYNAPTIC-MEMBRANES [J].

BOWERY, NG ;

HILL, DR ;

HUDSON, AL .

BRITISH JOURNAL OF PHARMACOLOGY, 1983, 78 (01) :191-206

[3] SIMPLE AND SENSITIVE SATURATION ASSAY METHOD FOR MEASUREMENT OF ADENOSINE 3'-5'-CYCLIC MONOPHOSPHATE [J].

BROWN, BL ;

ALBANO, JDM ;

EKINS, RP ;

SGHERZI, AM ;

TAMPION, W .

BIOCHEMICAL JOURNAL, 1971, 121 (03) :561-+

[4] THE SYNTHESIS OF PHOSPHONOBACLOFEN, AN ANTAGONIST OF BACLOFEN [J].

CHIEFARI, J ;

GALANOPOULOS, S ;

JANOWSKI, WK ;

KERR, DIB ;

PRAGER, RH .

AUSTRALIAN JOURNAL OF CHEMISTRY, 1987, 40 (09) :1511-1518

[5] GABA, BICUCULLINE AND CENTRAL INHIBITION [J].

CURTIS, DR ;

DUGGAN, AW ;

FELIX, D ;

JOHNSTON, GA .

NATURE, 1970, 226 (5252) :1222-&

[6]

DAWSON JM, 1984, ANAL BIOCHEM, V51, P429

[7] BICUCULLINE-INSENSITIVE GABA RECEPTORS - STUDIES ON THE BINDING OF (-)-BACLOFEN TO RAT CEREBELLAR MEMBRANES [J].

DREW, CA ;

JOHNSTON, GAR ;

WEATHERBY, RP .

NEUROSCIENCE LETTERS, 1984, 52 (03) :317-321

[8] A PHYSIOLOGICAL-ROLE FOR GABAB RECEPTORS IN THE CENTRAL NERVOUS-SYSTEM [J].

DUTAR, P ;

NICOLL, RA .

NATURE, 1988, 332 (6160) :156-158

[9]

FALCH E, 1986, J NEUROCHEM, V47, P898

[10] BACLOFEN-H-3 AND H-3-GABA BIND TO BICUCULLINE-INSENSITIVE GABA-B SITES IN RAT-BRAIN [J].

HILL, DR ;

BOWERY, NG .

NATURE, 1981, 290 (5802) :149-152

← 1 2 3 4 →