IMPORTANCE OF A NOVEL GABAA RECEPTOR SUBUNIT FOR BENZODIAZEPINE PHARMACOLOGY

被引:1265
作者
PRITCHETT, DB
SONTHEIMER, H
SHIVERS, BD
YMER, S
KETTENMANN, H
SCHOFIELD, PR
SEEBURG, PH
机构
[1] UNIV HEIDELBERG,ZMBH,NEUENHEIMER FELD 282,D-6900 HEIDELBERG,FED REP GER
[2] UNIV HEIDELBERG,INST NEUROBIOL,D-6900 HEIDELBERG,FED REP GER
关键词
D O I
10.1038/338582a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:582 / 585
页数:4
相关论文
共 31 条
  • [1] [H-3]-LABELED PROPYL BETA-CARBOLINE-3-CARBOXYLATE AS A SELECTIVE RADIOLIGAND FOR THE BZ1 BENZODIAZEPINE RECEPTOR SUBCLASS
    BRAESTRUP, C
    NIELSEN, M
    [J]. JOURNAL OF NEUROCHEMISTRY, 1981, 37 (02) : 333 - 341
  • [2] CASALOTTI SO, 1986, J BIOL CHEM, V261, P5013
  • [3] HIGH-EFFICIENCY TRANSFORMATION OF MAMMALIAN-CELLS BY PLASMID DNA
    CHEN, C
    OKAYAMA, H
    [J]. MOLECULAR AND CELLULAR BIOLOGY, 1987, 7 (08) : 2745 - 2752
  • [4] PYRAZOLOQUINOLINES - 2ND GENERATION BENZODIAZEPINE RECEPTOR LIGANDS HAVE HETEROGENEOUS EFFECTS
    COOPER, SJ
    KIRKHAM, TC
    ESTALL, LB
    [J]. TRENDS IN PHARMACOLOGICAL SCIENCES, 1987, 8 (05) : 180 - 184
  • [5] CONSTRUCTION AND CHARACTERIZATION OF AN ACTIVE FACTOR-VIII VARIANT LACKING THE CENTRAL 1/3 OF THE MOLECULE
    EATON, DL
    WOOD, WI
    EATON, D
    HASS, PE
    HOLLINGSHEAD, P
    WION, K
    MATHER, J
    LAWN, RM
    VEHAR, GA
    GORMAN, C
    [J]. BIOCHEMISTRY, 1986, 25 (26) : 8343 - 8347
  • [6] VARIOUS PROTEINS FROM RAT-BRAIN, SPECIFICALLY AND IRREVERSIBLY LABELED BY [H-3]FLUNITRAZEPAM, ARE DISTINCT ALPHA-SUBUNITS OF THE GABA BENZODIAZEPINE RECEPTOR COMPLEX
    FUCHS, K
    MOHLER, H
    SIEGHART, W
    [J]. NEUROSCIENCE LETTERS, 1988, 90 (03) : 314 - 319
  • [7] THE STRYCHNINE-BINDING SUBUNIT OF THE GLYCINE RECEPTOR SHOWS HOMOLOGY WITH NICOTINIC ACETYLCHOLINE-RECEPTORS
    GRENNINGLOH, G
    RIENITZ, A
    SCHMITT, B
    METHFESSEL, C
    ZENSEN, M
    BEYREUTHER, K
    GUNDELFINGER, ED
    BETZ, H
    [J]. NATURE, 1987, 328 (6127) : 215 - 220
  • [8] IMPROVED PATCH-CLAMP TECHNIQUES FOR HIGH-RESOLUTION CURRENT RECORDING FROM CELLS AND CELL-FREE MEMBRANE PATCHES
    HAMILL, OP
    MARTY, A
    NEHER, E
    SAKMANN, B
    SIGWORTH, FJ
    [J]. PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1981, 391 (02): : 85 - 100
  • [9] FUNCTIONAL MODULATION OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR BY TYROSINE PHOSPHORYLATION
    HOPFIELD, JF
    TANK, DW
    GREENGARD, P
    HUGANIR, RL
    [J]. NATURE, 1988, 336 (6200) : 677 - 680
  • [10] SELECTIVE ANTAGONISTS OF BENZODIAZEPINES
    HUNKELER, W
    MOHLER, H
    PIERI, L
    POLC, P
    BONETTI, EP
    CUMIN, R
    SCHAFFNER, R
    HAEFELY, W
    [J]. NATURE, 1981, 290 (5806) : 514 - 516