SYNTHESIS OF C-14-LABELED 1,4-BENZODIAZEPINES .4. C-13 AND C-14-LABELED 8-CHLORO-1-(2-DIMETHYLAMINO)ETHYL-6-PHENYL-4H-SIGMA-TRIAZOLO[4,3-A][1,4]-BENZODIAZEPINE TOSYLATE

被引：4

作者：

HSI, RSP

STOLLE, WT

机构：

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 1981年 / 18卷 / 06期

关键词：

D O I：

10.1002/jlcr.2580180613

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：881 / 888

页数：8

共 12 条

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[6] SYNTHESIS OF C-14-LABELED 1,4-BENZODIAZEPINES .3. 2-ALLYLOXY-AMINO-7-CHLORO-5-(2-CHLOROPHENYL)-3H-1,4-BENZODIAZEPINE-2-C-14, 8-CHLORO-1-DIMETHYLAMINO-METHYL-6-PHENYL-4H-S-TRIAZOLO[4,3-A][1,4]BENZODIAZEPINE-3A-C-14, AND 8-CHLORO-2,4-DIHYDRO-2-METHYL-6-PHENYL-1H-S-TRIAZOLO[4,3-A][1,4]BENZODIAZEPIN-1-ONE-3A-14 [J].

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JOHNSON, TD .

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[7] SYNTHESIS OF C-14-LABELED 1,4-BENZODIAZEPINES .1. 8-CHLORO-1-MEND 8-CHLORO-6-(2-CHLOROPHENYL)-1-METHYL-4H-S-TRIAZOLO[4,3-A] [1,ND 8-CHLORO-6-(2-CHLOROPHENYL)-1-METHYL-4H-S-TRIAZOLO[4,3-A] [1,4]BENZODIAZEPINE-1-C-14 [J].

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[9] BIOTRANSFORMATION OF 8-CHLORO-6-PHENYL-4H-S-TRIAZOLO[4,3-A] [1,4]BENZODIAZEPINE (D-40TA), A NEW CENTRAL DEPRESSANT, IN MAN, DOG AND RAT [J].

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[10] METABOLISM OF 8-CHLORO-6-(ORTHO-CHLOROPHENYL)-1-METHYL-4H-S-TRIAZOLO [4,3-A] [1,4]BENZODIAZEPINE, TRIAZOLAM, A NEW CENTRAL DEPRESSANT .2. IDENTIFICATION AND DETERMINATION OF METABOLITES IN RATS AND DOGS [J].

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