SPECIES-DIFFERENCES IN STRUCTURE-ACTIVITY-RELATIONSHIPS OF ADENOSINE AGONISTS AND XANTHINE ANTAGONISTS AT BRAIN ADENOSINE-A1-RECEPTORS

被引：79

作者：

UKENA, D

JACOBSON, KA

PADGETT, WL

AYALA, C

SHAMIM, MT

KIRK, KL

OLSSON, RO

DALY, JW

机构：

[1] NIDDKD,CHEM LAB,BETHESDA,MD 20892

[2] UNIV S FLORIDA,COLL MED,DEPT INTERNAL MED,TAMPA,FL 33612

来源：

FEBS LETTERS | 1986年 / 209卷 / 01期

关键词：

D O I：

10.1016/0014-5793(86)81096-1

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：122 / 128

页数：7

共 19 条

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[7] ADENOSINE RECEPTORS - TARGETS FOR FUTURE DRUGS [J].

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[8] ANALOGS OF CAFFEINE AND THEOPHYLLINE - EFFECT OF STRUCTURAL ALTERATIONS ON AFFINITY AT ADENOSINE RECEPTORS [J].

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[9] FUNCTIONALIZED CONGENERS OF ADENOSINE - PREPARATION OF ANALOGS WITH HIGH-AFFINITY FOR A1-ADENOSINE RECEPTORS [J].

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[10] [H-3] XANTHINE AMINE CONGENER OF 1,3-DIPROPYL-8-PHENYLXANTHINE - AN ANTAGONIST RADIOLIGAND FOR ADENOSINE RECEPTORS [J].

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DALY, JW .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (11) :4089-4093

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