CDPI3-ENEDIYNE AND CDPI3-EDTA CONJUGATES - A NEW CLASS OF DNA CLEAVING AGENTS

被引：62

作者：

BOGER, DL

ZHOU, JC

机构：

[1] Department of Chemistry, Scripps Research Institute, La Jolla, California 92037

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1993年 / 58卷 / 11期

关键词：

D O I：

10.1021/jo00063a019

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis and preliminary evaluation of la and lb, prototypical CDPI3-enediyne and CDPI3-EDTA conjugates constituting a new class of DNA cleaving agents, are detailed.

引用

页码：3018 / 3024

页数：7

共 64 条

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