PHARMACOKINETIC AND TUMOR-PENETRATION PROPERTIES OF THE HYPOXIC CELL RADIOSENSITIZER DESMETHYLMISONIDAZOLE (RO 05-9963) IN DOGS

被引:23
作者
WHITE, RAS [1 ]
WORKMAN, P [1 ]
机构
[1] MRC,CLIN ONCOL & RADIOTHERAPEUT UNIT,CAMBRIDGE,ENGLAND
关键词
D O I
10.1038/bjc.1980.39
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:268 / 276
页数:9
相关论文
共 17 条
  • [1] STRUCTURE-ACTIVITY-RELATIONSHIPS IN THE DEVELOPMENT OF HYPOXIC CELL RADIOSENSITIZERS .1. SENSITIZATION EFFICIENCY
    ADAMS, GE
    CLARKE, ED
    FLOCKHART, IR
    JACOBS, RS
    SEHMI, DS
    STRATFORD, IJ
    WARDMAN, P
    WATTS, ME
    PARRICK, J
    WALLACE, RG
    SMITHEN, CE
    [J]. INTERNATIONAL JOURNAL OF RADIATION BIOLOGY, 1979, 35 (02) : 133 - 150
  • [2] STRUCTURE-ACTIVITY-RELATIONSHIPS IN THE DEVELOPMENT OF HYPOXIC CELL RADIOSENSITIZERS .2. CYTOTOXICITY AND THERAPEUTIC RATIO
    ADAMS, GE
    CLARKE, ED
    GRAY, P
    JACOBS, RS
    STRATFORD, IJ
    WARDMAN, P
    WATTS, ME
    PARRICK, J
    WALLACE, RG
    SMITHEN, CE
    [J]. INTERNATIONAL JOURNAL OF RADIATION BIOLOGY, 1979, 35 (02) : 151 - 160
  • [3] ELECTRON-AFFINIC SENSITIZATION .7. CORRELATION BETWEEN STRUCTURES ONE-ELECTRON REDUCTION POTENTIALS, AND EFFICIENCIES OF NITROIMIDAZOLES AS HYPOXIC CELL RADIOSENSITIZERS
    ADAMS, GE
    FLOCKHART, IR
    SMITHEN, CE
    STRATFORD, IJ
    WARDMAN, P
    WATTS, ME
    [J]. RADIATION RESEARCH, 1976, 67 (01) : 9 - 20
  • [4] DISTRIBUTION OF MISONIDAZOLE IN HUMAN-TUMORS AND NORMAL-TISSUES
    ASH, DV
    SMITH, MR
    BUGDEN, RD
    [J]. BRITISH JOURNAL OF CANCER, 1979, 39 (05) : 503 - 509
  • [5] BROWN JM, 1978, BRIT J CANCER, V37, P206
  • [6] PHARMACOKINETIC CONSIDERATIONS IN TESTING HYPOXIC CELL RADIOSENSITIZERS IN MOUSE-TUMORS
    BROWN, JM
    YU, NY
    WORKMAN, P
    [J]. BRITISH JOURNAL OF CANCER, 1979, 39 (03) : 310 - 320
  • [7] CLINICAL TESTING OF RADIOSENSITIZER RO 07-0582 - EXPERIENCE WITH MULTIPLE DOSES
    DISCHE, S
    SAUNDERS, MI
    LEE, ME
    ADAMS, GE
    FLOCKHART, IR
    [J]. BRITISH JOURNAL OF CANCER, 1977, 35 (05) : 567 - 579
  • [8] FLOCKHART IR, 1978, BRIT J CANCER, V37, P264
  • [9] METABOLITE OF 2-NITROIMIDAZOLE MISONIDAZOLE WITH RADIOSENSITIZING PROPERTIES
    FLOCKHART, IR
    SHELDON, PW
    STRATFORD, IJ
    WATTS, ME
    [J]. INTERNATIONAL JOURNAL OF RADIATION BIOLOGY, 1978, 34 (01) : 91 - 94
  • [10] SAUNDERS MI, 1978, BRIT J CANCER, V37, P268