3-ALKYL-4-AMINOBUTYRIC ACIDS - THE 1ST CLASS OF ANTICONVULSANT AGENTS THAT ACTIVATES L-GLUTAMIC ACID DECARBOXYLASE

被引:78
作者
SILVERMAN, RB
ANDRUSZKIEWICZ, R
NANAVATI, SM
TAYLOR, CP
VARTANIAN, MG
机构
[1] NORTHWESTERN UNIV, INST NEUROSCI, EVANSTON, IL 60208 USA
[2] NORTHWESTERN UNIV, DEPT BIOCHEM MOLEC BIOL & CELL BIOL, EVANSTON, IL 60208 USA
[3] WARNER LAMBERT PARKE DAVIS, PARKE DAVIS PHARMACEUT RES DIV, DEPT PHARMACOL, ANN ARBOR, MI 48105 USA
关键词
D O I
10.1021/jm00111a053
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:2295 / 2298
页数:4
相关论文
共 48 条
[21]   EFFECT OF CONVULSIVE AGENT 3-MERCAPTOPROPIONIC ACID ON LEVELS OF GABA, OTHER AMINO-ACIDS AND GLUTAMATE DECARBOXYLASE IN DIFFERENT REGIONS OF RAT-BRAIN [J].
KARLSSON, A ;
FONNUM, F ;
MALTHESO.D ;
STORMMAT.J .
BIOCHEMICAL PHARMACOLOGY, 1974, 23 (21) :3053-3061
[22]  
Kodama K., 1981, SHINKEI KAGAKU, V20, P496
[23]  
LEWIS PJ, 1989, BR J CLIN PHARM S1, V27
[24]   BIOCHEMICAL CONSEQUENCES OF REACTIONS CATALYZED BY GAD AND GABA-T [J].
LIPPERT, B ;
JUNG, MJ ;
METCALF, BW .
BRAIN RESEARCH BULLETIN, 1980, 5 :375-379
[25]  
Lloyd KG, 1981, NEUROTRANSMITTERS SE, P325
[28]   VALPROATE ENHANCES GABA TURNOVER IN THE SUBSTANTIA NIGRA [J].
LOSCHER, W .
BRAIN RESEARCH, 1989, 501 (01) :198-203
[29]   REGIONAL ACTIVITIES OF METABOLIC ENZYMES AND GLUTAMATE-DECARBOXYLASE IN HUMAN-BRAIN [J].
MAKER, HS ;
WEISS, C ;
WEISSBARTH, S ;
SILIDES, DJ ;
WHETSELL, W .
ANNALS OF NEUROLOGY, 1981, 10 (04) :377-383
[30]  
McGeer E. G., 1983, GLUTAMINE GLUTAMATE, P3