THE BEHAVIOR OF INDENE OXIDE IN THE RITTER REACTION - A SIMPLE ROUTE TO CIS-AMINOINDANOL

被引：121

作者：

SENANAYAKE, CH

ROBERTS, FE

DIMICHELE, LM

RYAN, KM

LIU, J

FREDENBURGH, LE

FOSTER, BS

DOUGLAS, AW

LARSEN, RD

VERHOEVEN, TR

REIDER, PJ

机构：

[1] Merck Research Laboratories, Division of Merck, Co., Inc., Rahway, NJ 07065

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 23期

关键词：

D O I：

10.1016/0040-4039(95)00696-A

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A regio- and stereoselective synthesis of cis-1-aminoindan-2-ol via a Ritter reaction is described.

引用

收藏

页码：3993 / 3996

页数：4

相关论文

共 22 条

[1] HIGHLY DIASTEREOSELECTIVE REACTION OF A CHIRAL, NON-RACEMIC AMIDE ENOLATE WITH (S)-GLYCIDYL TOSYLATE - SYNTHESIS OF THE ORALLY-ACTIVE HIV-1 PROTEASE INHIBITOR L-735,524
ASKIN, D
ENG, KK
ROSSEN, K
PURICK, RM
WELLS, KM
VOLANTE, RP
REIDER, PJ
[J]. TETRAHEDRON LETTERS, 1994, 35 (05) : 673 - 676
[2] HIGHLY DIASTEREOSELECTIVE ALKYLATIONS OF CHIRAL AMIDE ENOLATES - NEW ROUTES TO HYDROXYETHYLENE DIPEPTIDE ISOSTERE INHIBITORS OF HIV-1 PROTEASE
ASKIN, D
WALLACE, MA
VACCA, JP
REAMER, RA
VOLANTE, RP
SHINKAI, I
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1992, 57 (10) : 2771 - 2773
[3] BACH RD, 1981, ORG SYNTH, V60, P63
[4] Bishop R., 1991, COMPREHENSIVE ORGANI, V6, P261
[5] CHEMICAL SYNTHESIS AND OPTICAL PURITY DETERMINATION OF OPTICALLY-ACTIVE 1,2-EPOXYINDAN AND ALCOHOL PRODUCTS WHICH ARE ALSO DERIVED FROM MAMMALIAN OR MICROBIAL-METABOLISM OF INDENE OR INDANONES
BOYD, DR
SHARMA, ND
SMITH, AE
[J]. JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1982, (11): : 2767 - 2770
[6] CHEMOENZYMATIC SYNTHESIS OF 1,2-AMINO-ALCOHOLS AND 1,3-AMINO-ALCOHOLS AND THEIR USE IN THE ENANTIOSELECTIVE REDUCTION OF ACETOPHENONE AND ANTI-ACETOPHENONE OXIME METHYL-ETHER WITH BORANE
DIDIER, E
LOUBINOUX, B
TOMBO, GMR
RIHS, G
[J]. TETRAHEDRON, 1991, 47 (27) : 4941 - 4958
[7] HALTERMAN RL, 1991, J ORG CHEM, V56, P5254
[8] HEATHCOCK C, 1967, J ORG CHEM, V32, P540
[9] JACOBSEN EN, 1994, CATALYTIC ASYMMETRIC, P159
[10] Krimen L. I., 1969, ORG REACTIONS, V17, P213, DOI DOI 10.1002/0471264180.0R017.03