DIFFERENCES IN THE INHIBITORY EFFECT OF CIMETIDINE ON DESIPRAMINE METABOLISM BETWEEN RAPID AND SLOW DEBRISOQUIN HYDROXYLATORS

被引:39
作者
STEINER, E [1 ]
SPINA, E [1 ]
机构
[1] HUDDINGE UNIV HOSP, METAB UNIT, S-14186 HUDDINGE, SWEDEN
关键词
D O I
10.1038/clpt.1987.147
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:278 / 282
页数:5
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共 31 条
  • [1] CIMETIDINE-INDUCED ALTERATIONS IN DESIPRAMINE PLASMA-CONCENTRATIONS
    AMSTERDAM, JD
    BRUNSWICK, DJ
    POTTER, L
    KAPLAN, MJ
    [J]. PSYCHOPHARMACOLOGY, 1984, 83 (04) : 373 - 375
  • [2] ROLE OF OXIDATION POLYMORPHISM ON BLOOD AND URINE CONCENTRATIONS OF AMITRIPTYLINE AND ITS METABOLITES IN MAN
    BALANTGORGIA, AE
    SCHULZ, P
    DAYER, P
    BALANT, L
    KUBLI, A
    GERTSCH, C
    GARRONE, G
    [J]. ARCHIV FUR PSYCHIATRIE UND NERVENKRANKHEITEN, 1982, 232 (03): : 215 - 222
  • [3] THE DEBRISOQUINE HYDROXYLATION TEST PREDICTS STEADY-STATE PLASMA-LEVELS OF DESIPRAMINE
    BERTILSSON, L
    ABERGWISTEDT, A
    [J]. BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1983, 15 (03) : 388 - 390
  • [4] HUMAN CYTOCHROMES-P-450
    BOOBIS, AR
    DAVIES, DS
    [J]. XENOBIOTICA, 1984, 14 (1-2) : 151 - 185
  • [5] BRENNAN RW, 1968, NEUROLOGY, V18, P283
  • [6] CRAMMER JL, 1969, PSYCHOPHARMACOLOGIA, V15, P207
  • [7] CIMETIDINE INTERACTION WITH AMITRIPTYLINE
    CURRY, SH
    DEVANE, CL
    WOLFE, MM
    [J]. EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1985, 29 (04) : 429 - 433
  • [8] CHARACTERIZATION OF A COMMON GENETIC-DEFECT OF CYTOCHROME-P-450 FUNCTION (DEBRISOQUINE-SPARTEINE TYPE POLYMORPHISM) - INCREASED MICHAELIS CONSTANT (KM) AND LOSS OF STEREOSELECTIVITY OF BUFURALOL 1'-HYDROXYLATION IN POOR METABOLIZERS
    DAYER, P
    GASSER, R
    GUT, J
    KRONBACH, T
    ROBERTZ, GM
    EICHELBAUM, M
    MEYER, UA
    [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 125 (01) : 374 - 380
  • [9] EFFECT OF OXIDATIVE POLYMORPHISM (DEBRISOQUINE SPARTEINE TYPE) ON HEPATIC 1ST-PASS METABOLISM OF BUFURALOL
    DAYER, P
    BALANT, L
    KUPFER, A
    STRIBERNI, R
    LEEMANN, T
    [J]. EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1985, 28 (03) : 317 - 320
  • [10] DELMILLER D, 1983, AM J PSYCHIAT, V140, P351