Structure-based design of sulfonamide-substituted non-peptidic HIV protease inhibitors

[1] BISHETEROARYLPIPERAZINE REVERSE-TRANSCRIPTASE INHIBITOR IN COMBINATION WITH 3'-AZIDO-3'-DEOXYTHYMIDINE OR 2',3'-DIDEOXYCYTIDINE SYNERGISTICALLY INHIBITS HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REPLICATION IN-VITRO [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1994, 38 (02) : 288 - 293

[2] Darke P L, 1994, Adv Pharmacol, V25, P399, DOI 10.1016/S1054-3589(08)60438-X

[3] A NOVEL NONPEPTIDE HIV-1 PROTEASE INHIBITOR - ELUCIDATION OF THE BINDING MODE AND ITS APPLICATION IN THE DESIGN OF RELATED ANALOGS [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (17) : 2664 - 2677

[4] MACROMODEL - AN INTEGRATED SOFTWARE SYSTEM FOR MODELING ORGANIC AND BIOORGANIC MOLECULES USING MOLECULAR MECHANICS [J]. JOURNAL OF COMPUTATIONAL CHEMISTRY, 1990, 11 (04) : 440 - 467

[5] PAPAIN I, 1967, BIOCHEM BIOPH RES CO, V27, P157

[6] PRADA JVN, 1995, J MED CHEM, V38, P898

[7] PRASAD JVNV, 1994, J AM CHEM SOC, V116, P6989

[8] REDSHAW S, 1994, EXPERT OPIN INV DRUG, V3, P273

[9] USE OF MEDIUM-SIZED CYCLOALKYL RINGS TO ENHANCE SECONDARY BINDING - DISCOVERY OF A NEW CLASS OF HUMAN-IMMUNODEFICIENCY-VIRUS (HIV) PROTEASE INHIBITORS [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (11) : 1884 - 1891

[10] STRUCTURE-BASED DESIGN OF NONPEPTIDIC HIV PROTEASE INHIBITORS FROM A CYCLOOCTYLPYRANONE LEAD STRUCTURE [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (22) : 4463 - 4473

[1] BISHETEROARYLPIPERAZINE REVERSE-TRANSCRIPTASE INHIBITOR IN COMBINATION WITH 3'-AZIDO-3'-DEOXYTHYMIDINE OR 2',3'-DIDEOXYCYTIDINE SYNERGISTICALLY INHIBITS HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REPLICATION IN-VITRO [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1994, 38 (02) : 288 - 293

[2] Darke P L, 1994, Adv Pharmacol, V25, P399, DOI 10.1016/S1054-3589(08)60438-X

[3] A NOVEL NONPEPTIDE HIV-1 PROTEASE INHIBITOR - ELUCIDATION OF THE BINDING MODE AND ITS APPLICATION IN THE DESIGN OF RELATED ANALOGS [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (17) : 2664 - 2677

[4] MACROMODEL - AN INTEGRATED SOFTWARE SYSTEM FOR MODELING ORGANIC AND BIOORGANIC MOLECULES USING MOLECULAR MECHANICS [J]. JOURNAL OF COMPUTATIONAL CHEMISTRY, 1990, 11 (04) : 440 - 467

[5] PAPAIN I, 1967, BIOCHEM BIOPH RES CO, V27, P157

[6] PRADA JVN, 1995, J MED CHEM, V38, P898

[7] PRASAD JVNV, 1994, J AM CHEM SOC, V116, P6989

[8] REDSHAW S, 1994, EXPERT OPIN INV DRUG, V3, P273

[9] USE OF MEDIUM-SIZED CYCLOALKYL RINGS TO ENHANCE SECONDARY BINDING - DISCOVERY OF A NEW CLASS OF HUMAN-IMMUNODEFICIENCY-VIRUS (HIV) PROTEASE INHIBITORS [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (11) : 1884 - 1891

[10] STRUCTURE-BASED DESIGN OF NONPEPTIDIC HIV PROTEASE INHIBITORS FROM A CYCLOOCTYLPYRANONE LEAD STRUCTURE [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (22) : 4463 - 4473