(D-ALA2,N-VAL5), (D-ALA2,MET5) ENKEPHALINS AND ENKEPHALINAMIDES - CORRELATION BETWEEN BIOLOGICAL-ACTIVITY AND NMR FEATURES

被引：9

作者：

GAIRIN, JE ^{[1
]}

HARAN, R ^{[1
]}

MAZARGUIL, H ^{[1
]}

AUDIGIER, Y ^{[1
]}

CROS, J ^{[1
]}

机构：

[1] UNIV TOULOUSE 3,CNRS,PHARMACOL & TOXIKOL LAB,F-31078 TOULOUSE,FRANCE

来源：

FEBS LETTERS | 1981年 / 128卷 / 01期

关键词：

D O I：

10.1016/0014-5793(81)81077-0

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：51 / 54

页数：4

共 20 条

[1] (D-ALA2,N-VAL5) ENKEPHALINAMIDE AND (D-MET2,N-VAL)5 ENKEPHALINAMIDE - 2 POTENT AGONISTS OF OPIATE AND ENKEPHALIN RECEPTORS [J].

AUDIGIER, Y ;

MAZARGUIL, H ;

CROS, J .

FEBS LETTERS, 1980, 110 (01) :88-90

[2]

AUDIGIER Y, 1980, EUR J MED CHEM, V15, P173

[3] STRUCTURE-ACTIVITY-RELATIONSHIPS OF ENKEPHALIN ANALOGS AT OPIATE AND ENKEPHALIN RECEPTORS - CORRELATION WITH ANALGESIA [J].

AUDIGIER, Y ;

MAZARGUIL, H ;

GOUT, R ;

CROS, J .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 63 (01) :35-46

[4]

BEDDELL CR, 1977, P R SOC LONDON B, V198, P229

[5] EXPERIMENTAL CALIBRATION OF A KARPLUS RELATIONSHIP IN ORDER TO STUDY CONFORMATIONS OF PEPTIDES BY NUCLEAR MAGNETIC-RESONANCE [J].

CUNG, MT ;

MARRAUD, M ;

NEEL, J .

MACROMOLECULES, 1974, 7 (05) :606-613

[6] CONFORMATIONAL-ANALYSIS OF LINEAR PEPTIDES BY N-15 NMR-SPECTROSCOPY USING THE ENKEPHALIN-RELATED FRAGMENT TYR-GLY-GLY-PHE AS A MODEL-COMPOUND [J].

GARBAYJAUREGUIBERRY, C ;

BAUDET, J ;

FLORENTIN, D ;

ROQUES, BP .

FEBS LETTERS, 1980, 115 (02) :315-318

[7] MODE OF DEACTIVATION OF ENKEPHALINS BY RAT AND HUMAN-PLASMA AND RAT-BRAIN HOMOGENATES [J].

HAMBROOK, JM ;

MORGAN, BA ;

RANCE, MJ ;

SMITH, CFC .

NATURE, 1976, 262 (5571) :782-783

[8] NMR-STUDY ON MET-ENKEPHALIN AND MET-ENKEPHALINAMIDE - MOLECULAR ASSOCIATION AND CONFORMATION [J].

HIGASHIJIMA, T ;

KOBAYASHI, J ;

NAGAI, U ;

MIYAZAWA, T .

EUROPEAN JOURNAL OF BIOCHEMISTRY, 1979, 97 (01) :43-57

[9] EFFECT OF MORPHINE ON ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS ASSESSMENT OF AGONIST AND ANTAGONIST POTENCIES OF NARCOTIC ANALGESICS [J].

HUGHES, J ;

KOSTERLITZ, HW ;

LESLIE, FM .

BRITISH JOURNAL OF PHARMACOLOGY, 1975, 53 (03) :371-381

[10] MOLECULAR-CONFORMATIONS OF MET-ENKEPHALIN - COMPARISON OF ZWITTERIONIC AND CATIONIC FORMS [J].

JONES, CR ;

GARSKY, V ;

GIBBONS, WA .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1977, 76 (03) :619-625

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