SYNTHESIS OF IODOALKYLACYLATES AND THEIR USE IN THE PREPARATION OF S-ALKYL PHOSPHOROTHIOLATES

被引：17

作者：

IYER, RP ^{[1
]}

YU, D ^{[1
]}

HO, NH ^{[1
]}

AGRAWAL, S ^{[1
]}

机构：

[1] TUFTS UNIV,DEPT CHEM,MEDFORD,MA 02155

来源：

SYNTHETIC COMMUNICATIONS | 1995年 / 25卷 / 18期

关键词：

D O I：

10.1080/00397919508011821

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Synthesis of iodoalkylacylates 3a-f and use of 3 c in the preparation of an oligonucleoside phosphorothiate prodrug analog 5 is described.

引用

页码：2739 / 2749

页数：11

共 20 条

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