MULTIPLE PATHWAYS OF PROPRANOLOLS METABOLISM ARE INHIBITED BY DEBRISOQUIN

被引:9
作者
ANTHONY, L [1 ]
KOSHAKJI, R [1 ]
WOOD, AJJ [1 ]
机构
[1] VANDERBILT UNIV,DEPT PHARMACOL,NASHVILLE,TN 37232
关键词
D O I
10.1038/clpt.1989.141
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:297 / 300
页数:4
相关论文
共 14 条
[1]   CRITICAL EVALUATION OF THE POTENTIAL ERROR IN PHARMACOKINETIC STUDIES OF USING THE LINEAR TRAPEZOIDAL RULE METHOD FOR THE CALCULATION OF THE AREA UNDER THE PLASMA LEVEL TIME CURVE [J].
CHIOU, WL .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1978, 6 (06) :539-546
[2]   CONTRIBUTION OF ENVIRONMENTAL-FACTORS TO VARIABILITY IN HUMAN DRUG-METABOLISM [J].
DOLLERY, CT ;
FRASER, HS ;
MUCKLOW, JC ;
BULPITT, CJ .
DRUG METABOLISM REVIEWS, 1979, 9 (02) :207-220
[3]   DEFECTIVE N-OXIDATION OF SPARTEINE IN MAN - NEW PHARMACOGENETIC DEFECT [J].
EICHELBAUM, M ;
SPANNBRUCKER, N ;
STEINCKE, B ;
DENGLER, HJ .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1979, 16 (03) :183-187
[4]   POLYMORPHIC OXIDATION OF SPARTEINE AND DEBRISOQUINE - RELATED PHARMACOGENETIC ENTITIES [J].
EICHELBAUM, M ;
BERTILSSON, L ;
SAWE, J ;
ZEKORN, C .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1982, 31 (02) :184-186
[5]  
GUENGERICH FP, 1986, MOL PHARMACOL, V30, P287
[6]   HUMAN-LIVER CYTOCHROMES-P-450 INVOLVED IN POLYMORPHISMS OF DRUG OXIDATION [J].
GUENGERICH, FP ;
DISTLERATH, LM ;
REILLY, PEB ;
WOLFF, T ;
SHIMADA, T ;
UMBENHAUER, DR ;
MARTIN, MV .
XENOBIOTICA, 1986, 16 (05) :367-378
[7]   IMPROVED HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC METHOD FOR THE SIMULTANEOUS DETERMINATION OF PROPRANOLOL AND 4-HYDROXYPROPRANOLOL IN PLASMA WITH FLUORESCENCE DETECTION [J].
KOSHAKJI, RP ;
WOOD, AJJ .
JOURNAL OF CHROMATOGRAPHY-BIOMEDICAL APPLICATIONS, 1987, 422 :294-300
[8]   PURIFICATION AND CHARACTERIZATION OF THE RAT-LIVER MICROSOMAL CYTOCHROME-P-450 INVOLVED IN THE 4-HYDROXYLATION OF DEBRISOQUINE, A PROTOTYPE FOR GENETIC-VARIATION IN OXIDATIVE DRUG-METABOLISM [J].
LARREY, D ;
DISTLERATH, LM ;
DANNAN, GA ;
WILKINSON, GR ;
GUENGERICH, FP .
BIOCHEMISTRY, 1984, 23 (12) :2787-2795
[9]   POLYMORPHIC HYDROXYLATION OF DEBRISOQUINE IN MAN [J].
MAHGOUB, A ;
IDLE, JR ;
DRING, LG ;
LANCASTER, R ;
SMITH, RL .
LANCET, 1977, 2 (8038) :584-586
[10]  
OTTON SV, 1988, DRUG METAB DISPOS, V16, P15