QUINOXALINE DERIVATIVES ARE HIGH-AFFINITY ANTAGONISTS OF THE NMDA RECEPTOR-ASSOCIATED GLYCINE SITES

被引：134

作者：

KESSLER, M

BAUDRY, M

LYNCH, G

机构：

来源：

BRAIN RESEARCH | 1989年 / 489卷 / 02期

关键词：

D O I：

10.1016/0006-8993(89)90875-5

中图分类号：

Q189 [神经科学];

学科分类号：

071006 ;

摘要：

引用

收藏

页码：377 / 382

页数：6

相关论文

共 28 条

[1] DIFFERENTIAL MODULATION OF [H-3]TCP BINDING TO THE NMDA RECEPTOR BY L-GLUTAMATE AND GLYCINE [J].

BENAVIDES, J ;

RIVY, JP ;

CARTER, C ;

SCATTON, B .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 149 (1-2) :67-72

[2] CNQX BLOCKS ACIDIC AMINO-ACID INDUCED DEPOLARIZATIONS AND SYNAPTIC COMPONENTS MEDIATED BY NON-NMDA RECEPTORS IN RAT HIPPOCAMPAL SLICES [J].

BLAKE, JF ;

BROWN, MW ;

COLLINGRIDGE, GL .

NEUROSCIENCE LETTERS, 1988, 89 (02) :182-186

[3]

BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3

[4] LIGHT MICROSCOPIC AUTORADIOGRAPHIC LOCALIZATION OF [H-3] GLYCINE AND [H-3] STRYCHNINE BINDING-SITES IN RAT-BRAIN [J].

BRISTOW, DR ;

BOWERY, NG ;

WOODRUFF, GN .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 126 (03) :303-307

[5] NEW QUINOXALINEDIONES SHOW POTENT ANTAGONISM OF QUISQUALATE RESPONSES IN CULTURED MOUSE CORTICAL-NEURONS [J].

DREJER, J ;

HONORE, T .

NEUROSCIENCE LETTERS, 1988, 87 (1-2) :104-108

[6] PHENCYCLIDINE AND RELATED DRUGS BIND TO THE ACTIVATED N-METHYL-D-ASPARTATE RECEPTOR CHANNEL COMPLEX IN RAT-BRAIN MEMBRANES [J].

FAGG, GE .

NEUROSCIENCE LETTERS, 1987, 76 (02) :221-227

[7] GLYCINE REVERSES ANTAGONISM OF N-METHYL-D-ASPARTATE (NMDA) BY 1-HYDROXY-3-AMINOPYRROLIDONE-2 (HA-966) BUT NOT BY D-2-AMINO-5-PHOPHONOVALERATE (D-AP5) ON RAT CORTICAL SLICES [J].

FLETCHER, EJ ;

LODGE, D .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 151 (01) :161-162

[8] THE NOVEL ANTICONVULSANT MK-801 BINDS TO THE ACTIVATED STATE OF THE N-METHYL-D-ASPARTATE RECEPTOR IN RAT-BRAIN [J].

FOSTER, AC ;

WONG, EHF .

BRITISH JOURNAL OF PHARMACOLOGY, 1987, 91 (02) :403-409

[9] 6,7-DICHLORO-3-HYDROXY-2-QUINOXALINECARBOXYLIC ACID IS A RELATIVELY POTENT ANTAGONIST AT NMDA AND KAINATE RECEPTORS [J].

FREY, P ;

BERNEY, D ;

HERRLING, PL ;

MUELLER, W ;

URWYLER, S .

NEUROSCIENCE LETTERS, 1988, 91 (02) :194-198

[10] QUINOXALINEDIONES - POTENT COMPETITIVE NON-NMDA GLUTAMATE RECEPTOR ANTAGONISTS [J].

HONORE, T ;

DAVIES, SN ;

DREJER, J ;

FLETCHER, EJ ;

JACOBSEN, P ;

LODGE, D ;

NIELSEN, FE .

SCIENCE, 1988, 241 (4866) :701-703