ENOL ESTERS AS INTERMEDIATES FOR THE FACILE CONVERSION OF AMINO-ACIDS INTO AMIDES AND DIPEPTIDES

被引：46

作者：

KABOUCHE, Z ^{[1
]}

BRUNEAU, C ^{[1
]}

DIXNEUF, PH ^{[1
]}

机构：

[1] UNIV RENNES 1,CNRS,CHIM COORDINAT ORGAN LAB,CAMPUS BEAULIEU,F-35042 RENNES,FRANCE

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 39期

关键词：

RUTHENIUM CATALYSIS; ENOL ESTERS; ALPHA-AMINO AMIDES; DIPEPTIDES;

D O I：

10.1016/S0040-4039(00)92385-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

N-Protected amino enol esters are easily transformed at room temperature into amino amides, and in the presence of potassium cyanide as catalyst, into tertiary amides and dipeptides.

引用

页码：5359 / 5362

页数：4

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