CHRONIC ADMINISTRATION OF MORPHINE AND NALTREXONE UP-REGULATE MU-OPIOID BINDING-SITES LABELED BY [H-3][D-ALA2,MEPHE4,GLY-OL5]ENKEPHALIN - FURTHER EVIDENCE FOR 2 MU-BINDING SITES

被引:91
作者
ROTHMAN, RB
BYKOV, V
LONG, JB
BRADY, LS
JACOBSON, AE
RICE, KC
HOLADAY, JW
机构
[1] NIDDK,NEUROL LAB,DRUG DESIGN & SYNTH SECT,BETHESDA,MD 20892
[2] WALTER REED ARMY INST RES,DIV NEUROPSYCHIAT,WASHINGTON,DC 20307
[3] NIMH,FUNCT NEUROANAT UNIT,BETHESDA,MD 20892
关键词
D O I
10.1016/0014-2999(89)90655-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:71 / 82
页数:12
相关论文
共 56 条
  • [1] EVALUATION OF THE INTERACTIONS OF MU AND DELTA SELECTIVE LIGANDS WITH [H-3]D-ALA2-D-LEU5-ENKEPHALIN BINDING TO MOUSE-BRAIN MEMBRANES
    BARRETT, RW
    VAUGHT, JL
    [J]. LIFE SCIENCES, 1983, 33 (24) : 2439 - 2448
  • [2] BROWN BMJ, 1977, STATISTICS BIOMEDICA, P118
  • [3] MULTIPLE OPIATE RECEPTORS - PHYLOGENETIC DIFFERENCES
    BUATTI, MC
    PASTERNAK, GW
    [J]. BRAIN RESEARCH, 1981, 218 (1-2) : 400 - 405
  • [4] PROBES FOR NARCOTIC RECEPTOR MEDIATED PHENOMENA .12. CIS-(+)-3-METHYLFENTANYL ISOTHIOCYANATE, A POTENT SITE-DIRECTED ACYLATING AGENT FOR SIGMA-OPIOID RECEPTORS - SYNTHESIS, ABSOLUTE-CONFIGURATION, AND RECEPTOR ENANTIOSELECTIVITY
    BURKE, TR
    JACOBSON, AE
    RICE, KC
    SILVERTON, JV
    SIMONDS, WF
    STREATY, RA
    KLEE, WA
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (06) : 1087 - 1093
  • [5] CHANG KJ, 1979, J BIOL CHEM, V254, P2610
  • [6] CONTRERAS PC, 1984, J PHARMACOL EXP THER, V229, P21
  • [7] Danks J A, 1986, NIDA Res Monogr, V75, P93
  • [8] CHRONIC ADMINISTRATION OF MORPHINE AND NALTREXONE UP-REGULATE[H-3][D-ALA2,D-LEU5]ENKEPHALIN BINDING-SITES BY DIFFERENT MECHANISMS
    DANKS, JA
    TORTELLA, FC
    LONG, JB
    BYKOV, V
    JACOBSON, AE
    RICE, KC
    HOLADAY, JW
    ROTHMAN, RB
    [J]. NEUROPHARMACOLOGY, 1988, 27 (09) : 965 - 974
  • [9] DECOSTA BR, IN PRESS J MED CHEM
  • [10] EVIDENCE FOR THE NEUROPEPTIDE CHOLECYSTOKININ AS AN ANTAGONIST OF OPIATE ANALGESIA
    FARIS, PL
    KOMISARUK, BR
    WATKINS, LR
    MAYER, DJ
    [J]. SCIENCE, 1983, 219 (4582) : 310 - 312