EVALUATION OF THE INTERACTIONS OF MU AND DELTA SELECTIVE LIGANDS WITH [H-3]D-ALA2-D-LEU5-ENKEPHALIN BINDING TO MOUSE-BRAIN MEMBRANES

被引:25
作者
BARRETT, RW [1 ]
VAUGHT, JL [1 ]
机构
[1] RUTGERS STATE UNIV,COLL PHARM,DEPT PHARMACOL & TOXICOL,PISCATAWAY,NJ 08854
关键词
D O I
10.1016/0024-3205(83)90638-0
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2439 / 2448
页数:10
相关论文
共 15 条
[1]   THE EFFECTS OF RECEPTOR SELECTIVE OPIOID-PEPTIDES ON MORPHINE-INDUCED ANALGESIA [J].
BARRETT, RW ;
VAUGHT, JL .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 80 (04) :427-430
[2]  
BARRETT RW, 1983, THESIS RUTGERS U
[3]  
CHANG KJ, 1979, J BIOL CHEM, V254, P2610
[4]   MORPHICEPTIN (NH4-TYR-PRO-PHE-PRO-CONH2) - A POTENT AND SPECIFIC AGONIST FOR MORPHINE (MU) RECEPTORS [J].
CHANG, KJ ;
KILLIAN, A ;
HAZUM, E ;
CUATRECASAS, P ;
CHANG, JK .
SCIENCE, 1981, 212 (4490) :75-77
[5]   [H-3]TYR-D-SER-GLY-PHE-LEU-THR - A SPECIFIC PROBE FOR THE DELTA-OPIATE RECEPTOR SUBTYPE IN BRAIN MEMBRANES [J].
DAVID, M ;
MOISAND, C ;
MEUNIER, JC ;
MORGAT, JL ;
GACEL, G ;
ROQUES, BP .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 78 (03) :385-387
[6]   COMPARISON OF THE BINDING CHARACTERISTICS OF TRITIATED OPIATES AND OPIOID-PEPTIDES [J].
GILLAN, MGC ;
KOSTERLITZ, HW ;
PATERSON, SJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 70 (03) :481-490
[7]   SPECTRUM OF THE MU-BINDING, DELTA-BINDING AND KAPPA-BINDING SITES IN HOMOGENATES OF RAT-BRAIN [J].
GILLAN, MGC ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 77 (03) :461-468
[8]   NALOXAZONE IRREVERSIBLY INHIBITS THE HIGH-AFFINITY BINDING OF [I-125]D-ALA2-D-LEU5-ENKEPHALIN [J].
HAZUM, E ;
CHANG, KJ ;
CUATRECASAS, P ;
PASTERNAK, GW .
LIFE SCIENCES, 1981, 28 (26) :2973-2979
[9]  
MUNSON PJ, 1980, ANAL BIOCH, V107, P1765
[10]  
OLIGIATI V, 1982, LIFE SCI, V31, P1675