ELECTROPHYSIOLOGICAL STUDIES WITH NEW CCK ANALOGS - CORRELATION WITH BINDING-AFFINITY ON B-TYPE RECEPTORS

被引:14
作者
BOHME, GA [1 ]
DURIEUX, C [1 ]
STUTZMANN, JM [1 ]
CHARPENTIER, B [1 ]
ROQUES, BP [1 ]
BLANCHARD, JC [1 ]
机构
[1] UER SCI PHARMACEUT & BIOL, INSERM, U266, CNRS, DEPT CHIM ORGAN, UA 498, F-7500L PARIS, FRANCE
关键词
D O I
10.1016/0196-9781(89)90051-X
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:407 / 414
页数:8
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共 57 条
  • [31] 2 BRAIN CHOLECYSTOKININ RECEPTORS - IMPLICATIONS FOR BEHAVIORAL ACTIONS
    MORAN, TH
    ROBINSON, PH
    GOLDRICH, MS
    MCHUGH, PR
    [J]. BRAIN RESEARCH, 1986, 362 (01) : 175 - 179
  • [32] INHIBITORY EFFECT OF CHOLECYSTOKININ OCTAPEPTIDE ON NEURONS IN THE NUCLEUS TRACTUS SOLITARIUS
    MORIN, MP
    DEMARCHI, P
    CHAMPAGNAT, J
    VANDERHAEGHEN, JJ
    ROSSIER, J
    DENAVITSAUBIE, M
    [J]. BRAIN RESEARCH, 1983, 265 (02) : 333 - 338
  • [33] RAPID APPEARANCE OF INTRAVENTRICULARLY ADMINISTERED NEUROPEPTIDES IN THE PERIPHERAL-CIRCULATION
    PASSARO, E
    DEBAS, H
    OLDENDORF, W
    YAMADA, T
    [J]. BRAIN RESEARCH, 1982, 241 (02) : 338 - 340
  • [34] [H-3] BOC [NLE28,31]CCK27-33, A NEW HIGHLY LABELED LIGAND FOR CCK RECEPTORS - BINDING ON BRAIN AND ON PANCREAS
    PELAPRAT, D
    ZAJAC, JM
    GACEL, G
    DURIEUX, C
    MORGAT, JL
    SASAKI, A
    ROQUES, BP
    [J]. LIFE SCIENCES, 1985, 37 (26) : 2483 - 2490
  • [35] AUTORADIOGRAPHY OF CCK RECEPTORS IN THE RAT-BRAIN USING [H-3] BOC[NLE28,31]CCK27-33 AND [I-125] BOLTON-HUNTER CCK8 - FUNCTIONAL-SIGNIFICANCE OF SUBREGIONAL DISTRIBUTIONS
    PELAPRAT, D
    BROER, Y
    STUDLER, JM
    PESCHANSKI, M
    TASSIN, JP
    GLOWINSKI, J
    ROSTENE, W
    ROQUES, BP
    [J]. NEUROCHEMISTRY INTERNATIONAL, 1987, 10 (04) : 495 - 508
  • [36] NEURONAL CHOLECYSTOKININ - ONE OR MULTIPLE TRANSMITTERS
    REHFELD, JF
    [J]. JOURNAL OF NEUROCHEMISTRY, 1985, 44 (01) : 1 - 10
  • [37] DISTRIBUTION OF NEUROPEPTIDES IN THE LIMBIC SYSTEM OF THE RAT - THE HIPPOCAMPUS
    ROBERTS, GW
    WOODHAMS, PL
    POLAK, JM
    CROW, TJ
    [J]. NEUROSCIENCE, 1984, 11 (01) : 35 - 77
  • [38] STUDIES ON THE CONFORMATION, ENZYMATIC DEGRADATION, PHARMACOLOGICAL POTENCY, AND BINDING-PROPERTIES IN BRAIN-TISSUE OF CHOLECYSTOKININ-8 AND NEW RELATED PEPTIDES
    ROQUES, BP
    DURIEUX, C
    GACEL, G
    PELAPRAT, D
    RUIZGAYO, M
    BELLENEY, J
    FELLION, E
    ZAJAC, JM
    FOURNIEZALUSKI, MC
    DAUGE, V
    MENANT, I
    ROSSIGNOL, P
    LUX, B
    GERARD, D
    BEGUE, D
    SASAKI, A
    MORGAT, JL
    [J]. ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1985, 448 (JUL) : 61 - 75
  • [39] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF BOC [NLE28, NLE31]CCK27-33, A HIGHLY POTENT CCK8 ANALOG
    RUIZGAYO, M
    DAUGE, V
    MENANT, I
    BEGUE, D
    GACEL, G
    ROQUES, BP
    [J]. PEPTIDES, 1985, 6 (03) : 415 - 420
  • [40] CHOLECYSTOKININ RECEPTORS IN THE BRAIN - CHARACTERIZATION AND DISTRIBUTION
    SAITO, A
    SANKARAN, H
    GOLDFINE, ID
    WILLIAMS, JA
    [J]. SCIENCE, 1980, 208 (4448) : 1155 - 1156