THE CONVERGENT SYNTHESIS OF CI-981, AN OPTICALLY-ACTIVE, HIGHLY POTENT, TISSUE SELECTIVE INHIBITOR OF HMG-COA REDUCTASE

被引：97

作者：

BAUMANN, KL ^{[1
]}

BUTLER, DE ^{[1
]}

DEERING, CF ^{[1
]}

MENNEN, KE ^{[1
]}

MILLAR, A ^{[1
]}

NANNINGA, TN ^{[1
]}

PALMER, CW ^{[1
]}

ROTH, BD ^{[1
]}

机构：

[1] CHEM DEPT,ANN ARBOR,MI 48105

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 17期

关键词：

D O I：

10.1016/S0040-4039(00)74190-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of Cl-981 is described starting from isobutyrylacetanilide (3) and the key chiral intermediate 2.

引用

页码：2283 / 2284

页数：2

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