THROMBOXANE SYNTHETASE INHIBITORS AS PHARMACOLOGICAL TOOLS - DIFFERENTIAL BIOCHEMICAL AND BIOLOGICAL EFFECTS ON PLATELET SUSPENSIONS

被引:60
作者
NEEDLEMAN, P
BRYAN, B
WYCHE, A
BRONSON, SD
EAKINS, K
FERRENDELLI, JA
MINKES, M
机构
[1] WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,ST LOUIS,MO 63110
[2] WASHINGTON UNIV,SCH MED,DEPT SURG,ST LOUIS,MO 63110
[3] COLUMBIA UNIV,COLL PHYS & SURG,NEW YORK,NY 10032
来源
PROSTAGLANDINS | 1977年 / 14卷 / 05期
关键词
D O I
10.1016/0090-6980(77)90306-9
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:897 / 907
页数:11
相关论文
共 25 条
[1]  
BUTCHER RW, 1962, J BIOL CHEM, V237, P1244
[2]   PROSTAGLANDIN ANTAGONISM BY SODIUM PARA-BENZYL-4-[1-OXO-2-(4-CHLOROBENZYL)-3-PHENYLPROPYL]PHENYLPHOSPHONATE (N-0164) [J].
EAKINS, KE ;
RAJADHYAKSHA, V ;
SCHROER, R .
BRITISH JOURNAL OF PHARMACOLOGY, 1976, 58 (03) :333-339
[3]   SELECTIVE INHIBITORY ACTIONS OF SODIUM-PARA-BENZYL-4-[1-OXO-2-(4-CHLOROBENZYL)-3-PHENYL PROPYL] PHENYL PHOSPHONATE (N-0164) AND INDOMETHACIN ON BIOSYNTHESIS OF PROSTAGLANDINS AND THROMBOXANES FROM ARACHIDONIC-ACID [J].
EAKINS, KE ;
KULKARNI, PS .
BRITISH JOURNAL OF PHARMACOLOGY, 1977, 60 (01) :135-140
[4]  
GORMAN R, IN PRESS
[5]   PROSTAGLANDIN-H1 AND PROSTAGLANDIN-H2 - CONVENIENT BIOCHEMICAL SYNTHESIS AND ISOLATION - FURTHER BIOLOGICAL AND SPECTROSCOPIC CHARACTERIZATION [J].
GORMAN, RR ;
SUN, FF ;
MILLER, OV ;
JOHNSON, RA .
PROSTAGLANDINS, 1977, 13 (06) :1043-1053
[6]  
GRYGLEWSKI RJ, NATURE, V267, P627
[7]   ISOLATION AND STRUCTURE OF 2 PROSTAGLANDIN ENDOPEROXIDES THAT CAUSE PLATELET-AGGREGATION [J].
HAMBERG, M ;
SVENSSON, J ;
WAKABAYASHI, T ;
SAMUELSSON, B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1974, 71 (02) :345-349
[8]   ISOMERIZATION OF PROSTAGLANDIN H-2 INTO PROSTAGLANDIN D2 IN PRESENCE OF SERUM-ALBUMIN [J].
HAMBERG, M ;
FREDHOLM, BB .
BIOCHIMICA ET BIOPHYSICA ACTA, 1976, 431 (01) :189-193
[9]  
HARPER JF, 1975, J CYCLIC NUCL PROT, V1, P207
[10]  
HASLAM R J, 1973, Series Haematologica, V6, P333