SYNTHESIS OF IMINOTHIASUGAR AS A POTENTIAL TRANSITION-STATE ANALOG INHIBITOR OF GLYCOSYLTRANSFER REACTIONS

被引：43

作者：

YUASA, H

KAJIMOTO, T

WONG, CH

机构：

[1] INST PHYS & CHEM RES, FRONTIER RES PROGRAM, GLYCOTECHNOL LAB, WAKO, SAITAMA 35101, JAPAN

[2] Scripps Res Inst, DEPT CHEM, LA JOLLA, CA 92037 USA

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 44期

关键词：

D O I：

10.1016/0040-4039(94)88293-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Iminothiasugar 1, a potential transition-state analog inhibitor of glycosidase

引用

页码：8243 / 8246

页数：4

共 12 条

[1] SYNTHESIS OF A BENZYLAMIDINE DERIVED FROM D-MANNOSE - A POTENT MANNOSIDASE INHIBITOR [J].

BLERIOT, Y ;

GENREGRANDPIERRE, A ;

TELLIER, C .

TETRAHEDRON LETTERS, 1994, 35 (12) :1867-1870

[2] NOVEL ROUTE TO 4-THIOFURANOSIDES - SYNTHESIS OF METHYL 4-THIO-ALPHA-D-TALOFURANOSIDE [J].

CLASSON, B ;

GAREGG, PJ ;

SAMUELSSON, B ;

LIU, ZC .

JOURNAL OF CARBOHYDRATE CHEMISTRY, 1987, 6 (04) :593-597

[3] SYNTHESIS OF OLIGOSACCHARIDES, GLYCOPEPTIDES, AND GLYCOLIPIDS [J].

HALCOMB, RL ;

WONG, CH .

CURRENT OPINION IN STRUCTURAL BIOLOGY, 1993, 3 (05) :694-700

[4] ENZYME-CATALYZED ALDOL CONDENSATION FOR ASYMMETRIC-SYNTHESIS OF AZASUGARS - SYNTHESIS, EVALUATION, AND MODELING OF GLYCOSIDASE INHIBITORS [J].

KAJIMOTO, T ;

LIU, KKC ;

PEDERSON, RL ;

ZHONG, ZY ;

ICHIKAWA, Y ;

PORCO, JA ;

WONG, CH .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1991, 113 (16) :6187-6196

[5]

Kanie O, 1992, CURR OPIN STRUC BIOL, V2, P674

[6] ENZYME-CATALYZED ORGANIC-SYNTHESIS - PRACTICAL ROUTES TO AZA SUGARS AND THEIR ANALOGS FOR USE AS GLYCOPROCESSING INHIBITORS [J].

LOOK, GC ;

FOTSCH, CH ;

WONG, CH .

ACCOUNTS OF CHEMICAL RESEARCH, 1993, 26 (04) :182-190

[7] DERIVATIVES OF 5-DEOXY-5-THIO-D-XYLOSE [J].

NESTADT, B ;

VANES, T .

TETRAHEDRON, 1968, 24 (04) :1973-&

[8]

PALCIC MM, 1989, J BIOL CHEM, V264, P17174

[9] ANTIBODY CATALYSIS OF GLYCOSIDIC BOND HYDROLYSIS [J].

REYMOND, JL ;

JANDA, KD ;

LERNER, RA .

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 1991, 30 (12) :1711-1713

[10] INHIBITION OF N-ACETYLGLUCOSAMINYLTRANSFER ENZYMES - CHEMICAL-ENZYMATIC SYNTHESIS OF NEW 5-MEMBERED ACETAMIDO AZASUGARS [J].

TAKAOKA, Y ;

KAJIMOTO, T ;

WONG, CH .

JOURNAL OF ORGANIC CHEMISTRY, 1993, 58 (18) :4809-4812

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