TOTAL SYNTHESIS OF DEPHOSTATIN, A NOVEL PROTEIN-TYROSINE-PHOSPHATASE INHIBITOR

被引：11

作者：

WATANABE, T

TAKEUCHI, T

OTSUKA, M

UMEZAWA, K

机构：

[1] KEIO UNIV,FAC SCI & TECHNOL,DEPT APPL CHEM,KOHOKU KU,YOKOHAMA 223,JAPAN

[2] INST MICROBIAL CHEM,SHINAGAWA KU,TOKYO 141,JAPAN

[3] KYOTO UNIV,INST CHEM RES,UJI,KYOTO 611,JAPAN

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1994年 / 04期

关键词：

D O I：

10.1039/c39940000437

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The first synthesis of dephostatin, conducted by use of a silyl protective group removable with HF-NaF buffer without damaging the labile N-nitrosamino group, is described.

引用

页码：437 / 438

页数：2

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