A CONVENIENT SYNTHESIS OF ALPHA',BETA-DIAMINO-ALPHA,ALPHA-DIFLUOROKETONES, NEW DIPEPTIDE ISOSTERES

被引：26

作者：

SCHIRLIN, D

BALTZER, S

ALTENBURGER, JM

机构：

来源：

TETRAHEDRON LETTERS | 1988年 / 29卷 / 30期

关键词：

D O I：

10.1016/S0040-4039(00)82154-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

收藏

页码：3687 / 3690

页数：4

相关论文

共 14 条

[1] ENZYME-INHIBITORS - GROUND-STATE TRANSITION-STATE ANALOGS
ABELES, RH
[J]. DRUG DEVELOPMENT RESEARCH, 1987, 10 (04) : 221 - 234
[2] CZERNECKI S, 1985, TETRAHEDRON LETT, P1699
[3] FEHRENTZ JA, 1983, SYNTHESIS-STUTTGART, P676
[4] FLUORO KETONE INHIBITORS OF HYDROLYTIC ENZYMES
GELB, MH
SVAREN, JP
ABELES, RH
[J]. BIOCHEMISTRY, 1985, 24 (08) : 1813 - 1817
[5] CONCEPT OF LINEAR MODIFIED RETRO-PEPTIDE STRUCTURES
GOODMAN, M
CHOREV, M
[J]. ACCOUNTS OF CHEMICAL RESEARCH, 1979, 12 (01) : 1 - 7
[6] 2,2-DIFLUORO-3-HYDROXYESTERS BY REFORMATSKII REACTION
HALLINAN, EA
FRIED, J
[J]. TETRAHEDRON LETTERS, 1984, 25 (22) : 2301 - 2302
[7] EXTENDED BINDING INHIBITORS OF CHYMOTRYPSIN THAT INTERACT WITH LEAVING GROUP SUBSITES S1'-S3'
IMPERIALI, B
ABELES, RH
[J]. BIOCHEMISTRY, 1987, 26 (14) : 4474 - 4477
[8] INHIBITION OF SERINE PROTEASES BY PEPTIDYL FLUOROMETHYL KETONES
IMPERIALI, B
ABELES, RH
[J]. BIOCHEMISTRY, 1986, 25 (13) : 3760 - 3767
[9] JUNG MYL, UNPUB
[10] KOLB M, 1988, UNPUB J MED CHEM