ELECTROPHILIC FLUORINATION IN THE SYNTHESIS OF NEW FLUOROINDOLES

被引：59

作者：

HODSON, HF

MADGE, DJ

SLAWIN, ANZ

WIDDOWSON, DA

WILLIAMS, DJ

机构：

[1] IMPERIAL COLL SCI TECHNOL & MED,DEPT CHEM,LONDON SW7 2AY,ENGLAND

[2] WELLCOME RES LABS,DEPT MED CHEM,BECKENHAM BR3 3BS,KENT,ENGLAND

[3] IMPERIAL COLL SCI TECHNOL & MED,CHEM CRYSTALLOG LAB,LONDON SW7 2AY,ENGLAND

来源：

TETRAHEDRON | 1994年 / 50卷 / 06期

关键词：

D O I：

10.1016/S0040-4020(01)80862-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Fluorination of trialkylstannylindoles with caesium fluoroxysulfate or Selectfluor(TM) was investigated for the synthesis of inter-alia 2- and 3-fluoroindoles. Caseium fluoroxysulfate gave good yields of these potentially useful intermediates; Selectfluor provided lower yields.

引用

页码：1899 / 1906

页数：8

共 25 条

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